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[(2-ethoxyphenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
3-(3-methyl-1H-pyrazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
3-{2-oxo-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}imidazolidine-2,4-dione
5-cyclopropyl-N-ethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(3-hydroxy-3-phenylpropyl)-N-methylacetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(oxolan-2-ylmethoxy)acetyl]piperidine-4-carboxylic acid
2-methyl-4-(4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}phenyl)butan-2-ol
2-{[2-(aminomethyl)piperidin-1-yl]methyl}-8-fluoroquinolin-4-ol
N-(2,4-dimethoxyphenyl)-3-[4-(2-hydroxyethyl)piperazin-1-yl]-3-oxopropanamide
4-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
7-(4-propylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-4H-pyran-2-carboxamide
1-{2-[(2-methylnaphthalen-1-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
2,4-dimethyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidine
1,3-dimethyl-6-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(5-{[(5-oxo-1-phenylpyrrolidin-3-yl)amino]methyl}furan-2-yl)benzonitrile
N'-(2-fluoro-5-methylphenyl)-N-[(3R)-oxolan-3-yl]butanediamide
N-methyl-5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(6-phenoxypyridin-3-yl)-1-(1-propylpiperidin-4-yl)piperidine-2-carboxamide
2-chloro-N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(2-ethylpyrimidin-5-yl)-N,3,6-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-[4-({[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]carbamoyl}methyl)phenyl]butanamide
2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-6-methylphenol
6-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(2-chlorophenyl)-3-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
2-(pyridin-2-ylmethyl)-9-[2-(pyrrolidin-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,5R)-5-[(dimethylamino)methyl]-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl]methanol
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(4-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperazin-2-one
1-[(3-fluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-6-oxopiperidine-3-carboxamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(quinolin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(3,3-diphenylpiperidin-1-yl)-3-oxopropyl]-N-methylmethanesulfonamide
3-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
8-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-5-(2-methylbenzenesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-cyclohexyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-benzyl-2-[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-(4,6-dimethylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propyl]piperidine-4-carboxamide
3-ethyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
2-[2-(dimethylamino)ethyl]-8-(quinoline-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]pyridine-2-carbonitrile
1-propyl-4-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-one
2-(4-methoxy-3-methylphenyl)-1-(pyrrolidin-3-ylmethyl)-1H-imidazole
2-({[(3R,4R)-4-(hydroxymethyl)-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4,6-difluoro-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(5-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}propanamide
2-(cyclohex-1-en-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one