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N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
2-[(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)methyl]benzoic acid
2-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
(2,4,6-trimethyl-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}phenyl)methanol
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
4-(4-{methyl[2-(4-methylphenoxy)ethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carbonitrile
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-(2-phenyl-1H-imidazol-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
N-({7-[2-(4-chloro-2-methylphenoxy)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
(2S)-2-amino-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentan-1-one
3-(furan-2-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-3-phenylpropan-1-one
3-fluoro-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
(2S,4R)-N-cyclopropyl-1-[(2-hydroxy-3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-amino-6-tert-butyl-4-(3-hydroxy-4-methoxyphenyl)pyridine-3-carbonitrile
(2S)-1-acetyl-N-(3-chloro-4-propanamidophenyl)pyrrolidine-2-carboxamide
1-[2-(4-fluorophenyl)ethyl]-4-{[(2E)-2-methylbut-2-en-1-yl]amino}pyrrolidin-2-one
1-methyl-4-({4-methyl-5-[1-(3-methylbutyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
1-(2-hydroxy-3-phenylpropyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N3-methyl-4-oxo-1-(2-phenylethyl)-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
(1S,3R)-3-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-3-ylmethyl)cyclopentane-1-carboxamide
N,N-dimethyl-4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
(1S,3R)-N-(oxan-4-yl)-3-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanamido]cyclopentane-1-carboxamide
2-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]benzene-1,3-diol
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2,4,5-trimethylbenzoyl)pyrrolidin-3-yl]acetamide
(3aR,7aS)-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1,5-dimethyl-3-(1H-pyrazol-3-yl)-1H-indazole
2,4-dimethoxy-6-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyrimidine
3-(4-fluorophenyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
5-chloro-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-[(5-methylthiophen-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[4-(1H-indol-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]pyridine-3-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2,6-dimethylquinoline
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(piperidin-4-ylmethyl)benzamide
1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(1-hydroxy-2-methylpropan-2-yl)piperidine-4-carboxamide
butyl N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
[2-(diethylamino)ethyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-3-(piperidin-1-yl)propan-1-one
1-cyclopentyl-3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-methylurea
N-[3-(1H-indazol-1-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-cyclopropyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(cyclohex-3-en-1-ylmethyl)piperidine-4-carboxamide
3-hydroxy-3-(2-methylphenyl)-N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]pyrrolidine-1-carboxamide
N-(4-methoxyphenyl)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-3-amine
({4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine