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2-[4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-1,3-benzoxazole
4-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-N-methylbenzene-1-sulfonamide
3-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-1H-indazole
7-methyl-2-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
1-({[1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyrrolidin-1-yl)ethyl]amine
2-(4-fluorophenyl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-[methyl(phenyl)amino]-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
2-[4-(1-ethoxyethyl)phenyl]-5-fluoropyridine
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-(2-fluorophenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(5-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl}-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
2-(furan-2-yl)-5-[1-(oxan-3-yl)-1H-imidazol-2-yl]pyrimidine
N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-4-(3-hydroxy-3-methylbutyl)benzamide
4-(1H-pyrazol-1-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidine-4-carboxylic acid
4-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
1-cyclohexyl-4-(4-oxo-4H-chromen-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-oxo-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
3-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,5,6-trimethyl-1,2-dihydropyridin-2-one
4-[(4-fluorophenyl)methyl]-N,N-dimethyl-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
4-{[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]methyl}morpholine
2-methoxy-4-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)pyridine-3-carbonitrile
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methoxyphenoxy)ethan-1-one
(1S,6R)-9-(1,3-benzothiazole-6-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
4-(hydroxymethyl)-N-[3-(methylsulfanyl)phenyl]-4-(2-phenylethyl)piperidine-1-carboxamide
4-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
7-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3S,4S)-1-(1-aminocyclobutanecarbonyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-chloro-N-(2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}ethyl)benzamide
3-[(3-propanamidophenyl)formamido]butanoic acid
(1-{2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethyl}piperidin-3-yl)methanol
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
1-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
2,4-dimethyl-N-(prop-2-en-1-yl)-N-propyl-1,3-thiazole-5-carboxamide
1-ethyl-4-[(3S)-3-ethylmorpholine-4-carbonyl]-1,2-dihydropyridin-2-one
1-{1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol
4-({1-[(2S)-2-aminopropanoyl]piperidin-4-yl}oxy)-3-chloro-N-(2-methoxyethyl)benzamide
N-{2-[4-phenyl-5-(pyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}aniline
2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxo-N-phenylacetamide
3-hydroxy-3-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
4-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
3-(3-fluorophenyl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-1H-pyrazole-4-carboxamide
(3aR,6aR)-2-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyrazin-2-yl)ethan-1-one
4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]thiomorpholine
N,8-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-{[3-(2-methylphenyl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate