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4-(dimethylsulfamoyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperazine-1-carboxamide
2-(5-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}furan-2-yl)benzonitrile
2-tert-butyl-4-hydroxy-N-[3-(1H-indazol-1-yl)propyl]pyrimidine-5-carboxamide
4-({3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
3-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
N-methyl-2-(2-methyl-1H-imidazol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
5-{1-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
2-(2-butyl-5-chloro-1H-imidazol-4-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(1S,5R)-3-(2,4-dimethylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methoxy-N-methyl-5-[({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}carbamoyl)amino]benzamide
(furan-2-ylmethyl)(1H-imidazol-4-ylmethyl)(3-methylbutan-2-yl)amine
3-(diphenylmethyl)-5-(3-methoxypropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(1-carbamoylcycloheptyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
2-(3-fluorophenyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
3-benzyl-8-(1H-imidazol-2-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-[(4-methyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-(propylsulfanyl)-1H-1,2,4-triazol-5-yl]acetamide
2-[2-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-4-(pyridin-2-yl)phenoxy]acetic acid
[(3,4-dimethoxyphenyl)methyl](methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-methyl-5-oxo-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-cyclopropyl-8-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
3-(2-chlorophenyl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
3-[5-(2-amino-6-methylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
4-[2-(propan-2-yl)-1H-imidazol-5-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1-benzylpyrrolidin-3-yl)-3-(1-cyclopropanecarbonylpiperidin-4-yl)propanamide
N3-[2-(4-ethoxyphenyl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1,2,3-thiadiazole-4-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidine
2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[1-(pyridin-4-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
4-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-thiazole-2-carboxamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(quinoxalin-2-yl)piperidin-3-ol
N-(1-cycloheptylpiperidin-3-yl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-3-yl}benzoic acid
2-hydroxy-1-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
(1R,2R)-N1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N2,N2-dimethyl-2,3-dihydro-1H-indene-1,2-diamine
7-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-3-(naphthalen-1-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(quinolin-3-ylmethyl)acetamide
N-ethyl-4-hydroxy-2-phenyl-N-(3-phenylpropyl)pyrimidine-5-carboxamide
4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]benzoic acid
3-(propan-2-yl)-5-[(2S)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
4-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{3-[(3-chlorophenyl)methyl]-1-phenylmethanesulfonylpiperidin-3-yl}methanol
3-{1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-N-methylpropanamide
2-(azepan-1-yl)-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}acetamide