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9-[2-(4-chlorophenoxy)ethyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-[(4aS,8aS)-7-(2,5-dimethylpyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N,N-dimethylacetamide
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methoxypyridine
N-tert-butyl-2-({[4-(2-methoxyphenoxy)phenyl]carbamoyl}amino)acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
5-(4-cyclohexylphenyl)-N-cyclopropyl-1,2,4-triazin-3-amine
2-(4-phenylpiperidin-1-yl)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-amino-4-methyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyrimidine-5-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-(2-hydroxy-2-phenylethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-(3-hydroxyphenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-2-one
N-(2-hydroxyethyl)-5-[1-(2-methylpropyl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2,4-dichlorophenoxy)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-1-[2-(azepan-1-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
6-(benzyloxy)-1-cyclohexyl-4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1,4-diazepan-2-one
1-cyclopentyl-5-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-chloro-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
1-{2-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
methyl (1R,3S,3aR,6aS)-3-[3-(4-chlorophenyl)-1H-pyrazol-4-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(2,5-dimethylphenyl)-N'-(2-hydroxyethyl)-N'-[(2E)-3-phenylprop-2-en-1-yl]propanediamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(2,3,6-trifluorophenyl)methyl]piperidine-4-carboxylate
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
(4aR,7aS)-1-(2-hydroxyethyl)-4-[4-(methylsulfanyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N4-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]pyrimidine-2,4-diamine
2-(4-propanoylphenoxy)-N-[2-(pyridin-2-yl)ethyl]acetamide
3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
2-{5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-(1H-1,3-benzodiazol-2-ylmethyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-cyclopropyl-1,3-oxazole-4-carboxamide
8-[2-(2-methylphenoxy)acetyl]-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-5-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}phenol
{[1-cyclohexyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}urea
2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(4-fluoro-2-methylphenyl)acetamide
3-[(3R,4S)-1-(6-aminopyridine-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(thiophen-2-ylmethyl)amine
2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methylphenol
N-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
N-(1-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
propan-2-yl 4-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amino}piperidine-1-carboxylate
2-(4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)-5-propylpyrimidine
1-(cyclohexylmethyl)-N3-ethyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[(1-phenylcyclopentyl)methyl]acetamide
2-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzonitrile