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(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
N-(1-{2-[4-(diphenylmethyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-fluorobenzamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
6-[benzyl(methyl)amino]-1-[(4-ethenylphenyl)methyl]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
7-fluoro-2-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-3-methyl-1H-indole
N-cyclopentyl-3,4,5-trimethoxy-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
(1R,5S)-6-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-6-azabicyclo[3.2.1]octane
2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)benzonitrile
methyl 2-[4-({[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]carbamoyl}amino)phenoxy]acetate
N-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1H-imidazol-2-ylmethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-2-yl)methyl]amine
(2S,4R)-4-amino-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
5-{4-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(2-methylbenzenesulfonyl)piperidine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[2-(3-fluorophenyl)ethyl]piperidine
1-cyclobutanecarbonyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]piperidine-4-carboxamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
4-{4-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-cyclohexanecarbonyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxamide
3-{1-[(3-chloro-1-benzothiophen-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-[(3-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(1-hydroxypropan-2-yl)benzamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-methanesulfonyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-[5-(azocan-1-ylmethyl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
6-(cyclopentylmethyl)-2-[4-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-(4-fluorophenyl)-N-(1H-imidazol-2-ylmethyl)-2-(piperidin-1-yl)acetamide
3-[2-(hydroxymethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
(4aS,8aR)-6-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
N-ethyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-ethyl-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine-3-carboxamide
1-[2-(dimethylamino)ethyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
7-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
1-(2,4-dimethylphenyl)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
2-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-chloro-N-(1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(3-hydroxypropyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
8-(4-ethyl-5-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 3-(2,6-dimethylpyrimidine-4-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{2-oxo-2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,N,4,5-tetramethyl-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-2-amine
N'-(3-chloro-4-methylphenyl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)propanediamide