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N-(6-fluoropyridin-3-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
2-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
2-{[(6-cyclopropylpyrimidin-4-yl)(methyl)amino]methyl}-2-ethylbutan-1-ol
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-methylpentan-1-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-hydroxyethyl)-2-propyl-N-(1,3-thiazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
(1S,6R)-3-methyl-9-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}morpholine
2-[5-(methoxymethyl)-1H-pyrazol-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3aR,7aS)-2-{2-[(6-ethoxypyridazin-3-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1-propyl-1H-pyrazole-5-carboxamide
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
2-(2-methoxyethyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}morpholine
1-cyclohexyl-4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-1,4-diazepane
3-{5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5-(1-benzofuran-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,2,4-triazin-3-amine
8-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3R,4R)-1-(2,5-dimethylbenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
3-chloro-5-{[3-(1,2-oxazolidine-2-carbonyl)-1,2-oxazol-5-yl]methoxy}pyridine
1-(2-methylpropyl)-2-phenylmethanesulfonyl-5-(pyrrolidin-1-ylmethyl)-1H-imidazole
N-({7-[4-(furan-2-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-indole-2-carboxamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[2-(morpholin-4-yl)ethyl]propanamide
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,3-oxazolidin-2-one
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-(2-fluorophenyl)-3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}propanamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propan-1-one
4-{3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4,6-dimethyl-2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethyl-4-(3-methylpiperidine-1-carbonyl)quinoline
1-[2-(benzyloxy)ethyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-[(3S,4R)-1-(5,6-dimethylpyrimidin-4-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-(2-methoxyethyl)-2-(2-oxopiperidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
({4-cyclopropyl-5-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(3R,5R)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2,3,6-trimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]quinoline-4-carboxamide
2-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]aniline
4-[(2-fluorophenyl)methyl]-3-oxo-N-(1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
8-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-methyl-5-{[4-phenyl-5-(2-phenylpropyl)-1H-imidazol-1-yl]methyl}pyrazine
1-(4-chloro-3-methylbenzoyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
ethyl 2-{[3-(thiophene-2-sulfonamidomethyl)piperidine-1-carbonyl]amino}acetate
6-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one