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1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-2-yl)ethan-1-one
methyl (2R,4S)-4-hydroxy-1-(2-methoxy-6-methylbenzoyl)piperidine-2-carboxylate
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(4aS,7aR)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{3-[ethyl(methyl)amino]-2-methylpropyl}-3-(1H-imidazol-2-yl)benzamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylpyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-amino-N,N-diethyl-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-2-carboxamide
N-(1-benzothiophen-2-ylmethyl)-2-(methoxymethyl)-N,6-dimethyl-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(3-methyl-4-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
(benzylsulfamoyl)(isoquinolin-5-ylmethyl)methylamine
6-(4-methoxyphenyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 1-(1H-imidazol-4-ylmethyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[2-(3,5-dimethylphenoxy)ethyl]-N,2-dimethyl-1,8-naphthyridine-3-carboxamide
4-methyl-3-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]benzamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(5-methylpyridine-3-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
5-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
6-[1-(2,5-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 3-benzamido-5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(methylsulfanyl)-N-(1,4-oxazepan-6-ylmethyl)pyrimidin-4-amine
4-{[(oxan-4-ylmethyl)carbamoyl]amino}-N-(2-phenylethyl)benzamide
4-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzamide
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
N-cyclopropyl-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazine-2-carboxamide
2-[(2-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
11-[2-(piperazin-1-yl)ethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-12-one
2-amino-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
[(3R,4R)-1-(1-benzofuran-5-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-ethyl-2-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
(3R,4R)-3-methyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-(oxan-4-yl)piperidin-4-ol
2-ethyl-5-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)pyrimidine
N-(2,3-dimethylphenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{1-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[2-methoxy-5-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
1-(3-chlorophenyl)-5-methyl-4-(4-methylbenzoyl)piperazin-2-one
1-(3-methoxyphenyl)-2,2-dimethyl-4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazine
6-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
1-cyclopropyl-N-[3-(1H-indol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
3-(methylsulfanyl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[3-(azepan-1-yl)-2-hydroxypropyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(4-chlorophenyl)-4-[(2,6-dimethoxyphenyl)methyl]morpholine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)acetamide