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7-fluoro-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]quinazolin-4-amine
7-oxo-N-[(1s,4s)-4-aminocyclohexyl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-3-sulfonamide
5-[(dimethylsulfamoyl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
N-cyclopentyl-N-[(2,3-dimethoxyphenyl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-[4-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(5-chloro-2-methoxybenzoyl)-1-(1,2-oxazol-3-ylmethyl)piperidine
2-[2-chloro-4-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)phenoxy]acetamide
1-ethyl-8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-fluoro-1-methyl-2-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-indole
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-2,3-dihydro-1H-isoindole-2-carboxamide
2-{1-benzyl-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(2,5-dimethylphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-methyl-5-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
N,N-diethyl-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
5-({[(3-{2-[4-(2,4-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-{3-cyclopropyl-5-[phenyl(1H-1,2,3,4-tetrazol-1-yl)methyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
N-methyl-N-(1-{[7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}pyrrolidin-3-yl)acetamide
3-{5-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
5-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N,N-dimethyl-4-(2-methyl-1-benzofuran-7-carbonyl)piperazine-1-sulfonamide
(2S)-2-{[3-(4-fluorophenyl)-1H-pyrazol-5-yl]formamido}-4-methylpentanamide
4-(1H-imidazol-1-yl)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidine-4-carboxylic acid
2-[1-(2,2-dimethylpropyl)-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazin-2-yl]ethan-1-ol
2-({[(3-chloro-4,5-diethoxyphenyl)methyl]amino}methyl)-3,5-dimethylpyridin-4-ol
(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
1-[(2-fluorophenyl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
(3S,5R)-N-ethyl-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carboxamide
1-(furan-2-ylmethyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidine-3-carboxamide
(3S,4R)-1-(2-cyclopentylacetyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(2-ethoxyethyl)-4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazole
2-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-imidazole
N-[4-(4-methylphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]pyridine-3-carboxamide
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(1-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(4-methylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-amino-3-ethyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(3-chlorophenyl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
1-cyclohexyl-3-(2-fluorophenyl)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-(pyridin-4-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
methyl 3-{imidazo[1,2-a]pyridine-2-carbonyl}-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one