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3-(dimethyl-1,2-oxazol-4-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
(3aS,6aS)-2-methanesulfonyl-5-[2-(pyridin-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyridine-4-carboxamide
(1R,2R,6S,7S)-4-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-(3-hydroxy-3-methylbutyl)-N-[3-(3-hydroxypiperidin-1-yl)propyl]benzamide
N-(oxolan-2-ylmethyl)-1-[1-(3-phenylprop-2-yn-1-yl)piperidin-4-yl]piperidine-4-carboxamide
6-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-[({[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-6-methyl-3,4-dihydropyrimidin-4-one
2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-1,3-thiazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
[1-(ethylsulfanyl)propan-2-yl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
[1-({methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclopropyl]methanol
7-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[(2,3-dihydro-1H-inden-2-yl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]thiophene-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-(3-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1S,6R)-9-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N,N,4-trimethyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}pyrimidin-2-amine
6-methyl-2-(7-methyl-1H-1,3-benzodiazol-2-yl)pyridin-3-ol
3-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methyl-5-sulfamoylphenyl)urea
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
[1-(2,4-dimethoxybenzoyl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
1-ethyl-4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N,5-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylpropanamido)benzamide
4-(1H-1,3-benzodiazol-1-yl)-1-(1,2-oxazole-3-carbonyl)piperidine-4-carboxylic acid
6-{[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
9-[(2-chloro-4-fluorophenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-2-oxo-8-[2-(propan-2-yl)pyrimidine-5-carbonyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{[4-(3,4-dimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
1-ethyl-5-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-ethyl-N-[2-(4-fluorophenyl)ethyl]-3-(hydroxymethyl)piperidine-1-carboxamide
4-({[(5-chlorofuran-2-yl)methyl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(pyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-{2-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
1-(propan-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
3,5-dichloro-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-4-methylbenzamide
methyl 3-({[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]carbamoyl}amino)-4-methylbenzoate
4-{1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-3-yl}benzoic acid
2-(3-chlorophenyl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
1-(cyclopropylmethyl)-3-hydroxy-3-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}piperidin-2-one
N-[3-(1H-indol-2-yl)phenyl]-1-(4-oxopentanoyl)piperidine-3-carboxamide
1-(3-hydroxyazetidin-1-yl)-2-[(3-methoxyphenyl)amino]butan-1-one
4-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
1-[4-({[2-(4-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol