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N-ethyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(methoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)cyclopropane-1-carboxamide
(3R,7S,8aS)-7-{[(2-chlorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(2S,4S)-4-(cyclooctylamino)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-ethyl-4-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
N-[3-(1H-indol-2-yl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-3-carboxamide
ethyl 1-{2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
2,2-dimethyl-N-{1-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
4-(2-{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-2-yl}ethyl)phenol
2-methyl-7-(oxane-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-benzyl-N5-ethyl-N3-methyl-4-oxo-N3-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-(2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-1-yl)acetic acid
2-methoxy-N-{2-methyl-3-[({2-[methyl(phenyl)amino]ethyl}carbamoyl)amino]phenyl}acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-N-[2-(pyridin-2-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-[(3,4-dimethoxyphenyl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-6-propylpyrimidine
N-[5-chloro-2-(2-methylpiperidin-1-yl)phenyl]-1H-1,2,4-triazole-5-carboxamide
methyl (2S,4R)-4-(2,4-dimethoxybenzamido)-1-[(2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
(2R,3R)-1'-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-benzyl-1-(isoquinoline-1-carbonyl)-N-methylpiperidin-3-amine
1-cyclopropanecarbonyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)piperidine-4-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichloro-4-methylbenzamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(2-oxo-1,3-oxazolidin-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(pyridin-4-yl)ethyl]-2-[(thiophen-2-ylmethyl)amino]benzamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-1-phenyl-1H-1,2,3-triazole
methyl 3-[(4-chlorophenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-5-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,8-dimethyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl (2S,4R)-4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamido]-1-methylpyrrolidine-2-carboxylate
N-propyl-7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[(2S,4R,6S)-2-ethyl-6-{2-phenylimidazo[1,2-a]pyridin-3-yl}oxan-4-yl]acetamide
2-(furan-2-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]azepane
3-[2-(4-fluorophenyl)ethyl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-N-ethylpiperidine-1-carboxamide
3-(azocan-1-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}propanamide
(3aS,6aS)-5-[(5-acetylthiophen-3-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-(morpholin-4-yl)ethane-1,2-dione
4-{[2-(2,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-2,6-dimethoxyphenol
2-methoxy-1-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepan-1-yl}ethan-1-one
7-(oxolane-2-amido)-N-(thiophen-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-{[1-(3-methoxyphenyl)propan-2-yl]amino}-N-(propan-2-yl)acetamide
1-(4-hydroxypiperidin-1-yl)-3-[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amine
N-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}-N-cyclopropyl-2,3-dimethoxybenzamide
1-(4-{4-[4-(2-methylpropyl)piperazin-1-yl]piperidin-1-yl}phenyl)pyrrolidin-2-one
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(propan-2-yl)pyrimidine-4-carboxamide