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8-{4-[1-(morpholin-4-yl)ethyl]phenyl}quinolin-4-amine
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
N-methyl-1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}pyrrolidine-3-carboxamide
3-[methyl({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})amino]propan-1-ol
N'-butyl-N'-[(2-fluorophenyl)methyl]-N,N-dimethylbutanediamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
9-(4-tert-butylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-3,4-dimethyl-1-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}pyrrolidin-3-ol
7-(cyclopropylmethyl)-2-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-1,2-oxazinane
2-methyl-4-(4-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}phenyl)butan-2-ol
2-[1-(2-fluorophenyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinolin-4-ol
4-[(8-hydroxyquinolin-2-yl)methyl]-1-methylpiperazine-2-carboxylic acid
3,5-dimethyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2-oxazole
2-[(4-chlorophenyl)sulfanyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-amino-4-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propylpyrimidine-5-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-ethylcyclopropyl)acetamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
ethyl 1-benzyl-5-{[4-(methoxycarbonyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(3-fluorophenyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-methyl-2-{5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-1H-imidazole
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
2-{2-[1-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
4-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
(2S,4R)-4-[2-(3,4-dimethylphenyl)acetamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
2-(1H-indol-3-yl)-N-(3-methoxypropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-(2-chlorophenyl)-N-[2-(4-hydroxyphenyl)ethyl]-2-methylfuran-3-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-(2-methoxyphenyl)-4-[4-(propan-2-yloxy)benzoyl]piperazin-2-one
2-{[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridin-6-yl]formamido}acetamide
3-[(dimethylamino)methyl]-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)pyrrolidin-3-ol
4-(piperidin-1-yl)-1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidine-4-carboxamide
(3aR,7aS)-2-(3-ethyl-1H-pyrazole-4-carbonyl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
[(3R,4R)-1-[4-(4-fluorophenyl)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
8-methoxy-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,N-dimethyl-5-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}pyrimidin-2-amine
1-(2-ethylbenzoyl)-2-(3-methoxypropyl)piperidine
(3aR,5R,6S,7aS)-2-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-octahydro-1H-isoindole-5,6-diol
3-methyl-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-carboxamide
2,5,6-trimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
3,5-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-{3-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}carbamoyl)methoxy]phenyl}propanamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-methyl-5-phenyl-N-[2-(propan-2-ylsulfanyl)ethyl]-1H-pyrazole-3-carboxamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole
(3aR,6aS)-5-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid