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1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-4-(pyridin-3-yl)piperidin-4-ol
4-benzyl-1-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]piperidine
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
(1R,5S)-3-(2-amino-6-methylpyrimidin-4-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{3-oxo-3-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
2-[(1S,5R)-6-(2,1,3-benzoxadiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-(2-methoxyethyl)-2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-(pyridin-3-ylmethyl)acetamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-[1-(thiophen-2-yl)ethyl]pyrrolidine-3-carboxamide
(1S,5R)-6-(1-methyl-1H-imidazole-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,5-dioxoimidazolidin-4-yl)-N-[3-(1H-indazol-1-yl)propyl]acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(1H-imidazol-1-yl)butanamide
[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
(1R,7S)-6-(4-acetyl-1,4-diazepane-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-ethyl-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxamide
2-(1H-indol-7-ylmethyl)-9-oxa-2-azaspiro[5.5]undecane
(4aR,7aS)-1-(2-methoxyethyl)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2,3-dihydro-1-benzofuran-7-carbonyl)-2-[(3-fluorophenyl)methyl]morpholine
{[5-(methoxymethyl)furan-2-yl]methyl}({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
4-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
3,4-dimethyl-N-[1-(pyridin-4-yl)propan-2-yl]-5-sulfamoylbenzamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-2,5-difluorobenzamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
1-[(2-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-benzyl-8-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
9-[(5-chlorothiophen-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,3R)-2-{[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-hydroxybutanamide
3-({1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
(1S,5R)-N-(2-ethylphenyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(4aR,8aS)-6-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
ethyl 5-(3-methoxy-3-oxopropyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{2-[2-(2,3,6-trimethylphenoxy)acetamido]ethyl}piperidine-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
2-(3-methoxyphenoxy)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
1-(pyridine-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
methyl 2-(2-{[2-(5-carbamoylthiophen-2-yl)pyrrolidin-1-yl]methyl}phenoxy)acetate
(2R,6S)-2,6-dimethyl-4-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]morpholine
N-[(2-methoxyphenyl)methyl]-N-propyl-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
(2S)-2-[(2,8-dimethylquinolin-4-yl)formamido]-3-(4-hydroxyphenyl)propanoic acid
3-ethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole-2-carboxamide
3-{5-[(3S)-3-hydroxy-3-phenylpropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 1-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidine-4-carboxylate
2-(morpholin-2-yl)-N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)acetamide
(2S,4R)-4-amino-1-(2-aminopyridine-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[(3-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)-N-(propan-2-yl)pentanamide