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(2S,4R)-4-amino-N,N-diethyl-1-[2-(2H-indazol-2-yl)acetyl]pyrrolidine-2-carboxamide
1-(2-aminopyrimidin-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[3-(3-methoxyphenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-7-methyl-1,2-dihydroquinolin-2-one
N,N,2-trimethyl-7-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(6-aminopyridine-3-carbonyl)-4-(2-hydroxyethyl)-1,4-diazepan-6-ol
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
6-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N,N-dimethylpyrazin-2-amine
4-({6-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridin-3-yl}methyl)morpholine
1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-({2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-N-methylpyridin-2-amine
4-(5-ethyl-1,2-oxazole-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
4-(1H-1,3-benzodiazol-2-yl)-2-chloro-6-methoxyphenol
2-methyl-6-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]-4H-pyran-4-one
2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)-6-methyl-1,2-dihydroquinolin-2-one
4-hydroxy-2-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]pyrimidine-5-carboxamide
1-(4-chlorophenyl)-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]cyclopropane-1-carboxamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-phenyl-5-[2-(propan-2-ylsulfanyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-cyclopropyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
1-[(5-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
7-[(2-methylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-fluoro-1-methyl-1H-indole
1-{5-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]thiophen-2-yl}ethan-1-one
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
N-(2,3-dihydro-1H-inden-2-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
5-{[3-(3,4-dimethylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}isoquinoline
3-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]-5-{[(3-methylphenyl)methyl]amino}benzamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(2-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenoxy)ethan-1-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]acetamide
1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-ol
1-(1-methyl-1H-pyrrol-2-yl)-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethane-1,2-dione
1-(3,4-dimethoxyphenyl)-3-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]urea
2-{4-[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]phenyl}-4,6-dimethoxypyrimidine
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(3R,4S)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(propan-2-yl)pyrrolidin-3-amine
N-[(3R,4R)-3-hydroxy-1-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}piperidin-4-yl]pyrazine-2-carboxamide
3,4,4-trimethyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidin-3-ol
N-[2-(azepane-1-carbonyl)phenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-(dimethylamino)-2-methylpropanamide
1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-benzyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
4-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-(naphthalen-1-yl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazine