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N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,3,5-trimethyl-1H-indole-2-carboxamide
2-{2-[(2,3-dihydroxypropyl)(methyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
8-fluoro-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]quinoline-2-carboxamide
1-(3-phenylpropyl)-5-(1H-pyrrole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S)-1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-ol
N-[(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-8-methoxyquinoline
(3R,4S)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-cyclopropyl-N,N-dimethylpyrrolidin-3-amine
2-methyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazole
(1S,5R)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(piperidin-1-ylmethyl)benzamide
4-{[methyl(1-methylpyrrolidin-3-yl)carbamoyl]amino}-N-(2-phenylethyl)benzamide
(3S,7S)-5-[4-(methylcarbamoyl)pyridin-2-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(3-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-3-oxopropyl)methanesulfonamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(1,3-thiazol-2-yl)ethyl]amino}methyl)piperidin-2-one
N-[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]-2-(pyrrolidin-3-yl)acetamide
2-[4-(piperidine-1-carbonyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(9H-purin-6-yl)piperidin-3-yl]propanamide
(1-{4-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]phenyl}ethyl)dimethylamine
N,N-dimethyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
3-(benzyloxy)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)azetidine
(2R,3R,6R)-5-(1H-indole-2-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-3-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]sulfamoyl}benzamide
2-(4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
3-[6-amino-5-cyano-4-(2-ethylpyrimidin-5-yl)pyridin-2-yl]benzoic acid
5-({methyl[(3-{2-[4-(2-phenylacetyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
(3aS,6aS)-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-chloro-3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
(1S,2R)-2-{[(6-methoxypyridin-3-yl)methyl](methyl)amino}cyclohexan-1-ol
2-(3,4-dimethoxyphenyl)-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2E)-2-methylbut-2-en-1-yl]amine
1-(2-benzylmorpholin-4-yl)-2-(diethylamino)ethan-1-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
2-(naphthalen-2-yl)-5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
5-fluoro-N4,N4-dimethyl-N2-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
(2R,6R)-4-(3-hydroxypyridine-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(cyclohexylmethyl)-5-[(2-methoxyethyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[4-(morpholin-4-ylmethyl)phenyl]urea
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)benzamide
2-ethyl-4-methyl-5-{3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-oxazole
(oxolan-2-ylmethyl)({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(thiophen-3-ylmethyl)amine
3-butyl-1-methyl-4-(thiophen-3-ylmethyl)piperazin-2-one
1-[(1R,5R)-6-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-N-propyl-3-(4H-1,2,4-triazol-4-yl)benzamide
N-cyclopropyl-4-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]sulfamoyl}benzamide
2-oxo-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(5-tert-butyl-1H-pyrazol-3-yl)methyl]({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine