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(1R,3S)-3-{[2-(4-fluorobenzenesulfonyl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]furan-2-carboxamide
(3S,5S)-1-benzyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[4-(dimethylamino)phenyl]methyl}pyrrolidin-3-amine
N-cyclopropyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide
ethyl 1-(2,5-difluorobenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-methyl-1-phenylurea
2-(dimethylamino)-N-[1-(hydroxymethyl)cyclopentyl]-2-(2-methylphenyl)acetamide
1'-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
4-(2-fluorophenoxy)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
2-(furan-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)azepane
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetamido]-N-(2-ethylphenyl)benzamide
(3S,4S)-4-cyclopropyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
2-(1H-1,2,3-benzotriazole-5-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4-fluorophenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1H-1,2,3-triazole-4-carboxamide
1-(morpholin-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]cyclohexane-1-carboxamide
1-(3-fluoropropyl)-4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
3-{4-[5-(hydroxymethyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
3-{[1-(piperidine-1-sulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
(3R,9R)-11-(4-ethylbenzoyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
6-cyclopentyl-3-{[(4-hydroxy-4-methylpentan-2-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
[3-(3-methylbut-2-en-1-yl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-3-yl]methanol
5-methyl-4-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-3-yl}-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(3-methylbutyl)azepan-4-amine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-cycloheptyl-1-(4-{[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(dimethylamino)ethyl]acetamide
3-[6-(morpholin-4-yl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
2-chloro-N-[2-(propane-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
8-(6-aminopyridine-3-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
11-{2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
2-(1H-1,2,4-triazol-1-ylmethyl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
4-{2-methyl-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-2-yl}morpholine
1,4,6-trimethyl-2-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-[(3S,4R)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
6-chloro-2-methyl-N-[(3R)-piperidin-3-yl]quinoline-4-carboxamide
1-(dimethylsulfamoyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-methylpropanamide
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
3-acetyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
[4-({4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide