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3-[(3-hydroxypiperidin-1-yl)methyl]-N-(quinoxalin-6-yl)benzamide
N-[2-(5-methoxyfuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
2-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[(3-methoxyphenyl)amino]butan-1-one
2-[4-(4-amino-5-methylpyrimidin-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-(3-fluorophenoxy)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
1-cyclohexyl-N-[(2,6-difluoro-3-methoxyphenyl)methyl]piperidine-4-carboxamide
N-ethyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
(3S,4R)-1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
6-methyl-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
(1S,5R)-6-(cyclobutylmethyl)-3-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-oxo-2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}ethyl)acetamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-{1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]azetidin-3-yl}pyridine
5-cyclopropanecarbonyl-1'-(5-fluoropyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclohexyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(prop-2-yn-1-yl)benzamide
4-({1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)morpholine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1-(propan-2-yl)cyclopropyl]acetamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{2-oxo-2-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
9-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(5-{[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
6-(3-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
6-({[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-N-[(1-hydroxycyclohexyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]thiomorpholine-4-carboxamide
(4aS,8aR)-6-[2-(3-methoxyphenyl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
2-methyl-6-[2-(pyridin-3-yloxy)propyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
methyl 2-{[2-(3-fluorophenyl)piperidine-1-carbonyl]amino}acetate
N4-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(3-fluorophenyl)-5-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)ethan-1-ol
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
N-[4-(2-fluorophenoxy)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
3-(3-methoxyphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
(2S)-4-(methylsulfanyl)-2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]butan-1-ol
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-{3-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-3-oxopropyl}-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
N-[4-(morpholin-4-yl)butan-2-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(2R,6R)-4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(3-methoxypropyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(cyclopropylmethyl)-3-(isoquinolin-5-yl)-6-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
propan-2-yl 4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-butyl-N-methyl-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide