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N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-amine
2-(3,5-difluorophenyl)-4-(1H-imidazol-1-ylmethyl)-5-methyl-1,3-oxazole
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-phenylethyl)piperidine
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-hydroxypropan-1-one
4-ethyl-6-(4-methanesulfonylphenyl)-2-(piperidin-1-yl)pyrimidine
N-[(6-chloropyridin-3-yl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
ethyl 4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-amido}piperidine-1-carboxylate
5-[(4-ethylpiperazin-1-yl)methyl]-N-(2-hydroxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-cyclopropyl-1-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-N-(3,5-dimethoxyphenyl)propanamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-5-methyl-2-phenyl-1H-imidazole
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]propan-1-ol
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
N-(2-methoxyethyl)-3-{1-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperidin-4-yl}propanamide
1-[3-({[(2-chlorophenyl)methyl]amino}methyl)-7-methylquinolin-2-yl]piperidin-4-ol
methyl 5-[(2,2-dimethylpropyl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carboxamide
7-amino-4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-(5-methyl-1,3-oxazole-4-carbonyl)-2-(2-phenylethyl)piperidine
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3-methyl-3-phenylpiperidine
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(furan-2-yl)propan-1-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1-propylpiperidin-4-amine
diethyl({3-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
(1R,5R)-6-benzyl-3-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
{1-[3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]piperidin-3-yl}methanol
1-[(2-chlorophenyl)methyl]-4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-4-yl)pyridine
5-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-indole-2-carboxamide
(3R,9aR)-3-benzyl-8-[(2,5-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(2-aminoacetyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-oxo-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(pyrrolidin-1-ylmethyl)pyrrolidine
1-(morpholin-4-yl)-2-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenoxy)ethan-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[1-(pyridin-4-yl)propyl]benzamide
2-(dimethylamino)-2-(4-methylphenyl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}ethan-1-one
7-(5-phenyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(3-chlorobenzoyl)-N-(3-methoxyphenyl)piperidine-1-carboxamide
3-(2-oxo-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)imidazolidine-2,4-dione
2-ethyl-5-{4-phenyl-1-[4-(pyridin-2-yl)butyl]-1H-imidazol-5-yl}pyrimidine
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-(propan-2-yl)piperazine
2-methyl-2-(1H-pyrrol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-hydroxypiperidine-4-carboxylic acid
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2,3,4-trimethoxybenzamide
3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-phenylpiperidine-1-carboxamide