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4-[2-(4-fluorophenyl)-2-hydroxyacetyl]-1-(2-methoxyphenyl)piperazin-2-one
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(prop-2-en-1-yl)acetamide
3,3-dimethyl-1-{[5-(quinolin-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
(2S)-2-amino-4-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}butanoic acid
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
methyl 1-[(3R,5S)-1-[(2-ethoxyphenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-phenyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}benzonitrile
6-[3-(piperidine-1-carbonyl)phenyl]-1,2,3,4-tetrahydroquinazoline-2,4-dione
4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3,3-dimethylpiperazin-2-one
6-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)-4-(trifluoromethyl)benzamide
8-(2,3-dimethylquinoxaline-6-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
5-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[1-(pyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2S,4S)-4-[4-({[(3,4-dimethylphenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N,N-dimethyl-4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-sulfonamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-[(2S)-2,3-dihydroxypropyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
3-{5-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-methyl-5-(2-{2-[(quinolin-4-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
methyl 1-(3-methylbutoxy)-8-[(3-methylquinoxalin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
9-[(2-methoxyphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(3-fluorophenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(5-chloropyridin-2-yl)-4-[4-(furan-2-yl)benzoyl]piperazine
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-phenyl-1H-pyrazole-4-carboxamide
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]propanamide
4-[(3-chlorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,5,6-trimethylpyrimidin-4-amine
3,3-dimethyl-1-({5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
4-[1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-3-yl]benzoic acid
2-(3-methoxypropyl)-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[2-(pyrrolidin-1-yl)ethyl]-1-(thiophene-3-sulfonyl)piperidine
(4aR,8aR)-2-cyclobutanecarbonyl-7-(4-methylphthalazin-1-yl)-decahydro-2,7-naphthyridin-4a-ol
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
1-(4-methylphenyl)-4-[3-(1H-pyrazol-1-yl)propanoyl]piperazin-2-one
N-cyclohexyl-6-oxo-N-(prop-2-yn-1-yl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(6-chloropyridazin-3-yl)-2-[(3-methoxyphenyl)methyl]morpholine
N-(1-{2-[4-(3-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
2-(2-hydroxyethyl)-8-(1-methyl-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-hydroxy-6-methylpyridin-2-yl)-3-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
N-cyclopropyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]benzene-1-sulfonamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{9-hydroxy-1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-3-yl}ethan-1-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1,3-diphenyl-1H-pyrazole-5-carboxamide
ethyl 1-(2-acetamidoacetyl)-3-(2-phenylethyl)piperidine-3-carboxylate