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4-[(2-methoxyethyl)(methyl)sulfamoyl]-N-(2-oxopyrrolidin-3-yl)benzamide
1-[(2-methoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
3-(azepane-1-carbonyl)-5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
1-{4-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,4-triazole
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]benzamide
2-(2,4-difluorophenyl)-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
2-(4-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(3-methoxypropyl)-1-methyl-5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]butanamide
N-[(3-chlorophenyl)methyl]-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidine
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yl)ethan-1-one
(2R,3S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylpentanamide
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
3-{5-[2-(1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridine-3-carboxamide
N-cyclopropyl-1-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
3-[(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
4-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
(1R,5S,6R)-3-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N,N-dimethyl-2-(4-{[4-(5-methylfuran-2-yl)phenyl]methyl}-1,4-diazepan-1-yl)acetamide
1-[5-methoxy-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
{1-[3-(3,5-dimethoxyphenyl)phenyl]ethyl}dimethylamine
4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpyridine-3-carboxamide
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N-cyclopentyl-4-oxobutanamide
ethyl 4-[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)amino]piperidine-1-carboxylate
3-{2-[ethyl({[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})amino]-1-hydroxyethyl}phenol
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2-fluorophenyl)-4-({3-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)piperazine
2,5-dimethyl-3-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrazine
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
(3aR,6aR)-2-[(3,4-dimethylphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-phenylethyl)-1-(1,3-thiazole-4-carbonyl)piperidine
(1S,5R)-3-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(5-chlorothiophen-2-yl)sulfonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
2-[4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)morpholin-3-yl]acetic acid
5-(4-fluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1,2,4-triazin-3-amine
2-methyl-5-[2-(2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}ethyl)morpholin-4-yl]-2,3-dihydropyridazin-3-one
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
2-(3-fluorophenyl)-2-hydroxy-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
5-[4-(2-ethoxyethyl)piperazine-1-carbonyl]quinoxaline
4-[(3-hydroxypiperidin-3-yl)methyl]-N-(2-methylphenyl)piperazine-1-carboxamide
N-[1-({[phenyl(pyridin-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide
N-[2-(benzyloxy)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide