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4-(1H-pyrazol-1-yl)-1-(quinoline-5-carbonyl)piperidine-4-carboxylic acid
(2S,4R)-4-amino-N-ethyl-1-(3-ethyl-1H-indole-2-carbonyl)pyrrolidine-2-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
2-(2-fluorophenyl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-{2,8-diazaspiro[4.5]decan-3-ylformamido}ethyl)-4-fluorobenzamide
3-(1H-indol-3-yl)-1-(3-propylmorpholin-4-yl)propan-1-one
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(3-methoxyphenyl)methyl]piperidine-4-carboxamide
1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-butyl-4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methylpiperazin-2-one
3-({4-[2-(4-chloro-2-methylphenoxy)ethyl]piperazin-1-yl}methyl)piperidin-3-ol
N-benzyl-N-(cyclobutylmethyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
N4,N4,N6-trimethyl-N6-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-4,6-diamine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pent-4-enamide
N,5-dimethyl-1-propyl-N-(quinolin-2-ylmethyl)-1H-pyrazole-4-carboxamide
3-(2-methylphenyl)-3-phenyl-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
3-{3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
(5S,9aS,9bS)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N,N-bis(2-hydroxyethyl)-5-methyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
methyl 4-(5-{[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
2-(3-methoxypropyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
1-(2-fluorobenzoyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-chloro-5-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-methyl-5-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-1-[(3-methylphenyl)methyl]piperazin-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-{spiro[2.4]heptane-1-carbonyl}piperidine-4-carboxamide
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazole
N-methyl-N-[2-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)ethyl]-3-phenylpropanamide
2-fluoro-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5-sulfamoylbenzamide
4-[5-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)furan-2-yl]-2-methylbut-3-yn-2-ol
(3S,4S)-1-[(2-methoxypyrimidin-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-(2-methoxyethyl)-N,1-dimethyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-{1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
2-[2-(2-chloro-4-fluorophenyl)phenyl]-5-methyl-1,3,4-oxadiazole
N-(1-benzothiophen-2-ylmethyl)-N-methyl-2-(3-methyl-2-oxoimidazolidin-1-yl)acetamide
4-(hydroxymethyl)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-ol
4-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
3-{[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
8-(3,5-dichloro-2-methoxybenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
4-(1H-pyrazol-1-yl)-2-[4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]butan-2-ol
4-(1H-imidazol-1-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}butan-1-one
3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
N-benzyl-2-[4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide