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1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-5-(1H-indazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-[1-(4-methanesulfonylphenyl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-(piperazin-1-yl)propan-2-ol
3-[3-(1-methoxyethyl)phenyl]-6-(4-methylpiperazin-1-yl)pyridazine
2-(2H-indazol-2-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-{[(6-cyclopropylpyrimidin-4-yl)amino]methyl}benzene-1-sulfonamide
1-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazole
3-cyclopentaneamido-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)benzamide
1-(3-cyanopyridin-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-(furan-3-yl)-6,8-dimethoxy-4-methylquinoline
3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1-(3-methylbut-2-en-1-yl)-1H-pyrazole
ethyl 2-{2-[(1-cyclopropyl-6-oxopiperidin-3-yl)formamido]ethyl}-1,3-thiazole-4-carboxylate
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
N-[1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)pyrrolidin-3-yl]acetamide
4-chloro-2-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
3-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazol-5-amine
N-[(1-methylpiperidin-2-yl)methyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
4-[(3,5-difluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-6-{5-[1-(1H-pyrrol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)acetamide
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[4-(morpholin-4-yl)butan-2-yl]propanamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
N-[1-(1H-imidazol-1-yl)propan-2-yl]-3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-amine
1-[2-(4-chlorophenyl)ethyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,4-dimethyl-5-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
7-(cyclobutylmethyl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[(4-methylphenyl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-(6-hydroxy-6-methylheptan-2-yl)-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
5-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}piperidin-2-one
5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridine-2-carbonitrile
2-{[4-(3-fluoro-2-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(3-methylcinnolin-5-yl)urea
6-(3-hydroxypiperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-{[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-3-chloropyridine
1-(cyclopropylmethyl)-5-(1H-indol-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-amino-6-(3,5-dimethylphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
9-[(4-chloro-3-fluorophenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methoxyphenyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1,2,4-oxadiazole
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
N-[3-(1H-indol-1-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
ethyl 4-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate