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(1S,6R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
7-(5-chloropyridin-2-yl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,4-dimethyl-5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,3-thiazol-2-amine
dimethyl[(5-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
2-(3,3-dioxo-1,3λ6,4-oxathiazinan-4-yl)-N-[2-(4-methoxyphenyl)ethyl]acetamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
2-benzyl-N-[2-(2-methylpropoxy)phenyl]-3-oxopiperazine-1-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl})methylamine
1-{2-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
7-(4-fluorophenyl)-2-(5-methyl-1,3,4-oxadiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[4-(2-methoxyphenyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
9-[(4-ethylphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2,2-dimethyl-1-(3-methylthiophen-2-yl)cyclopropanecarbonyl]piperazin-2-one
(3aR,5R,6S,7aS)-2-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydro-1H-isoindole-5,6-diol
1-[(2,3-dichloro-6-fluorophenyl)methyl]azepan-2-one
2-methyl-4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-oxazepane
3-(2-methoxyphenyl)-6-[4-(1H-pyrazol-1-yl)phenyl]pyridazine
N-methyl-2-(methylsulfanyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
2-(3-methyl-1H-pyrazol-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
1-[(1-{[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
(4aS,7aR)-1-(2-aminoacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-ethoxyphenyl)-N'-[1-(4-fluorophenyl)-2-methylpropan-2-yl]propanediamide
4-(1-benzyl-1H-pyrazol-4-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,2,3,6-tetrahydropyridine
6-ethyl-N-(1-methanesulfonylpiperidin-4-yl)-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(ethoxymethyl)-7-(1H-imidazol-4-ylmethyl)-N-(2-methylprop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(propan-2-yl)-1-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-4-methoxyphenol
ethyl 4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-1H-pyrazole-3-carboxylate
(1R,5S)-6-({5-[(dimethyl-1,2-oxazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-azabicyclo[3.2.1]octane
[(2E)-2-methylbut-2-en-1-yl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
1-benzyl-5-(1H-imidazol-4-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-N-(pyridin-2-ylmethyl)acetamide
2-(benzyloxy)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-methyl-2-{2-oxo-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(2-phenylpropan-2-yl)acetamide
N-(2H-1,3-benzodioxol-5-yl)-3-(2-methoxybenzoyl)piperidine-1-carboxamide
3-{2-amino-4-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-6-methylpyrimidin-5-yl}propanoic acid
1-(4-ethoxy-2-fluorophenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-{3-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2-methylphenyl}furan-2-carboxamide
N-benzyl-N-methyl-3-{[(oxan-4-yl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]ethan-1-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1-methyl-1H-pyrazole-5-carboxamide
2-hydroxy-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(methylsulfanyl)butan-1-one
N4-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(4-fluorophenyl)methyl]-4-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}piperazin-2-one
1-(2-fluorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]cyclopropane-1-carboxamide
N-(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}azepan-4-yl)methanesulfonamide