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2-(2-methoxy-5-methylphenyl)-1,3-benzoxazole
[1-(2-methyl-4-phenylpyridine-3-carbonyl)-3-propylpiperidin-3-yl]methanol
4-benzyl-3-ethyl-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-5-one
5-(2H-1,3-benzodioxol-4-ylmethyl)-1-(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{imidazo[1,2-a]pyridin-2-ylmethyl}[4-(1H-indol-3-yl)butan-2-yl]amine
1-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
2,3-dimethyl-5-phenyl-N-[2-(pyrazin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
8-fluoro-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-benzoyl-1-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
2-ethyl-5-fluoro-1-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
1-benzyl-3-(2-methoxyethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[5-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)furan-2-yl]methanol
4-[(6-methylpyridin-3-yl)oxy]-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidine-4-carboxylic acid
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
5-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-1H-1,2,3-benzotriazole
(1S,3R)-3-amino-N-[2-(4-chlorophenoxy)ethyl]-N-ethylcyclopentane-1-carboxamide
2-(4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
methyl 3-({[1-(4-chlorophenyl)cyclopropyl]formamido}methyl)-5-(furan-2-amido)benzoate
4-benzyl-3-methyl-1-{2-oxo-2-[2-(trifluoromethyl)pyrrolidin-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methoxy-5-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
(4-{[methyl({[3-(5-methylfuran-2-yl)phenyl]methyl})amino]methyl}oxan-4-yl)methanol
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
N-cyclopropyl-3-(2-methoxyphenyl)-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}propanamide
2-fluoro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
1-cyclohexyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}thiophene-3-sulfonamide
N-cyclopentyl-1-[1-(quinoxalin-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}pyridine
2-{3-cyclopropyl-5-[1-(prop-2-en-1-ylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
5-{1-[(3-methylthiophen-2-yl)sulfonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
{3-[2-methoxy-6-(4-phenyl-1H-imidazol-5-yl)phenoxy]propyl}dimethylamine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
2-amino-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-6-(4-methoxyphenyl)pyridine-3-carbonitrile
N3-[(4-ethoxyphenyl)methyl]-N3-(2-methoxyethyl)piperidine-1,3-dicarboxamide
1-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}cyclopentan-1-amine
4-chloro-1-methyl-3-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-indazole
4-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-3-yl}propanamide
2-{1-[(3,4-difluorophenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(1-benzothiophen-3-yl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(4-{1-[N-methyl-1-(1-methyl-1H-pyrazol-3-yl)formamido]-2-phenylethyl}piperidine-1-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylmorpholine-2-carboxamide
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(3,4-dimethoxyphenyl)acetic acid