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1-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazol-3-yl)phenol
dimethyl({2-[(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]ethyl})amine
4-benzyl-3-ethyl-1-[2-(pyridin-2-yl)ethyl]-1,4-diazepan-5-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,3-dihydroxypropyl)-1H-pyrazole-3-carboxamide
4-(3-chloro-5-fluorobenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-(3,5-dimethoxyphenyl)-3-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}propanamide
1-{1-[2-(propan-2-yloxy)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-(2-methyl-1-benzofuran-7-yl)piperidine-1-carboxamide
4-(5-chloro-2-methylphenyl)-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-amine
2-(4-fluorophenoxymethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1,3-oxazole-4-carboxamide
(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
5,6-dimethyl-2-oxo-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
({4-ethyl-5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
[4-(quinolin-2-yl)phenyl]methanol
8-(3,5-dichloropyridin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylquinoxaline-6-carboxamide
8-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-8-azaspiro[4.5]decane-7,9-dione
N-(3,5-dimethoxyphenyl)-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methyl-2-(pyrrolidin-1-yl)pyrimidine
2-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
2-[4-(dimethylamino)phenyl]-N-[(1-methylpiperidin-4-yl)methyl]acetamide
2-[1-(2,3-dimethylphenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
1-(cyclohexylmethyl)-N-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2,2-dimethylcyclopropyl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
3-(4-fluorophenyl)-4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-2-one
1-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-{[4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methyl}-4-(2-fluorophenyl)piperazine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-2-yl)acetamide
2-[3-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-[(3S,4R)-1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-[2-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
8-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
1-(2-fluorophenyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
2,3-dimethyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
5-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-2-hydroxybenzoic acid
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(pyridin-3-yloxy)propyl]pyridin-2-amine
5-(2H-1,3-benzodioxol-5-yl)-1-methyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole
1-[(5-{[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,4-dimethylphenyl)methyl]-1H-1,2,4-triazole
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxo-4-phenylbutanamide
6-(aminomethyl)-2-(4-ethoxyphenoxymethyl)-3,4-dihydropyrimidin-4-one
N-[1-(2-methoxyethyl)-7-[2-(2-methoxyethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
5-methyl-1-propyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-4-carboxamide
6-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one