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N-[1-(methoxymethyl)cyclopentyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
N-{1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}acetamide
(2R,6S)-4-[6-(3-chlorophenyl)-3-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]pyridin-2-yl]-2,6-dimethylmorpholine
(3S,4S)-4-cyclopropyl-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(methylsulfanyl)phenyl]methyl}amine
1-methyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}azepane-2-carboxamide
N-[2-(3-methylthiophen-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-methoxy-1-{1'-[2-(1-methylpiperidin-2-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-(pyridin-4-ylmethyl)urea
2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}morpholine-2-carboxamide
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]acetamide
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
8-fluoro-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(naphthalen-1-yl)-4H-1,2,4-triazole
4-chlorophenyl (7S,9aR)-7-ethyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-benzyl-N-[2-(dimethylamino)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-[2-(3-fluorophenyl)ethyl]-N-[3-(1H-imidazol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
1-cyclopentyl-N-[(2-methylphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-(furan-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidine-4-carboxamide
N-(pyridin-3-ylmethyl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
2-{[4-(3-{2-azabicyclo[2.2.1]heptan-2-yl}propanoyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
4-methyl-2-[4-(oxane-2-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
3-(1H-1,3-benzodiazol-2-yl)-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]propanamide
(3S,4R)-1-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-1-ethylpiperidine-2-carboxamide
N4-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-N2,6-dimethylpyrimidine-2,4-diamine
5-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(pyridin-2-ylmethyl)pyridin-2-amine
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
(4aR,7aS)-1-acetyl-4-(2-methoxy-3-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methylphenyl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-4-carboxamide
N-cyclopentyl-2-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propanamide
1-({1-[6-(2-fluorophenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-3,5,7-trimethyl-1H-indole
N-(oxolan-3-yl)-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
1,3-dimethyl-5-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
3-(1-benzyl-1H-imidazol-2-yl)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidine
3-(1-methyl-1H-pyrrol-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1H-pyrazole-5-carboxamide
6-(1-acetylpiperidine-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one