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1-(2,3-dihydro-1H-inden-2-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(methoxymethyl)pyrimidine
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(2-phenylethyl)piperidine
N-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}methanesulfonamide
1-(pyridin-4-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-(2-chloro-6-fluorophenyl)-1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[(3R,4S)-1-(4-cyanooxane-4-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-methyl-4-{[4-(piperidin-3-yl)phenyl]formamido}butanamide
5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[2-(3-methylthiophen-2-yl)ethyl]pyridin-2-amine
(3R,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-methoxyethyl)-N-methyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
methyl 2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}butanoate
2,4-dimethoxy-6-[4-(2,2,6,6-tetramethylpiperidin-4-yl)piperazin-1-yl]-1,3,5-triazine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
2-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-6-methylpyridine-3-carboxylic acid
1-{2-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
(3aR,6aR)-2-benzyl-5-(cyclopropanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,N-dimethyl-3-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)pyridin-2-amine
N,1-dimethyl-N-{1-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-3-carboxamide
4-[3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]morpholine
N,N-dimethyl-5-[({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)methyl]furan-2-carboxamide
N-[(3-chlorophenyl)methyl]-2-methyl-N-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrazine
6-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
5-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
2-(1H-imidazol-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
1-(2-{[(dicyclopropylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
6-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-(1H-imidazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl}acetamide
3-({[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}(pyridin-4-ylmethyl)amino)propan-1-ol
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-(oxan-4-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-(3-hydroxypropyl)-8-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1,3,4-oxadiazol-2-amine
(3S,4R)-1-(1H-indazole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-(2-methoxyethyl)-N3-[(2-methoxyphenyl)methyl]-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
6-(2-chlorophenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-hydroxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
1-(2-{[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)imidazolidin-2-one
[2-({4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}methyl)phenyl]methanol
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-ethylpyrimidine-5-carboxamide
2-(3-cyano-3-methylpiperidine-1-carbonyl)thiophene-3-sulfonamide
1-[2-(3-methoxyphenyl)azetidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[(3-fluoro-4-methylphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile