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N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
5-methanesulfonyl-N-[(5-methylpyrazin-2-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
N-methyl-5-[({[2-(piperidin-1-ylmethyl)phenyl]carbamoyl}amino)methyl]furan-2-carboxamide
11-[bis(prop-2-en-1-yl)amino]-4-[(2-methoxyphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(1R,5S,8R)-3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
3-[(4aR,7aS)-6,6-dioxo-4-[3-(pyrrolidin-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(2-butoxybenzoyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
2,7-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-fluoro-N,2-dimethyl-N-(1,2-oxazol-5-ylmethyl)quinoline-4-carboxamide
N-[2-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
{4-[(3,5-dichloropyridin-4-yl)methyl]morpholin-2-yl}methanamine
N-({1-[(3,7-dimethyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
6-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]pyrimidine-2,4-diamine
1-[4-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[2-(3-chlorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-(3-methylpyridin-4-yl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-diazepane
(3S,4S)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-ethyl-5-oxo-N-[(3-phenoxyphenyl)methyl]pyrrolidine-3-carboxamide
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(pyrrolidin-1-yl)propan-1-one
4-(2-phenylethyl)-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazole
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
3-(3-fluorophenyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
(4aS,8aR)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
6-fluoro-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-ol
1-[4-(ethylsulfanyl)phenyl]-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
N-{[5-(3-methylpyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl]sulfamoyl})amine
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]acetamide
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-[3-(4H-1,2,4-triazol-4-yl)propyl]urea
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(4-hydroxyphenyl)methyl]-5-methylpiperidin-2-one
2-benzyl-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,8-diazaspiro[5.5]undecane
N-benzyl-4-({4-[(3-hydroxypyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
1-butyl-5-(1H-imidazol-1-ylmethyl)-3-(phenoxymethyl)-1H-1,2,4-triazole
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
1-ethyl-5-[(oxan-4-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(1-cyclohexyl-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
5-(cyclopropylmethyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
1-(2,3-dihydro-1H-inden-4-yl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
4-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1-oxaspiro[4.4]nonan-2-one
(1R,2S,6R,7S)-4-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
6-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-propylpyridine-3-carboxamide
N-(2-methylphenyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine-1-carboxamide