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9-(3-fluoropyridin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
2-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}furan-2-yl)-1-methyl-1H-1,3-benzodiazole
1-methyl-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyrazin-2-amine
9-[(2-aminopyridin-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(pyrrolidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,5-dimethyl-1H-pyrazol-4-yl)-3-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}urea
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(2-fluoropyridin-3-yl)-3-methylurea
3-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-N,N-dimethylaniline
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(1-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)(quinolin-4-ylmethyl)amine
N-(5,6-dimethyl-1H-1,3-benzodiazol-7-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(1S,3R)-N-[(2-fluorophenyl)methyl]-3-(3-methanesulfonamidopropanamido)cyclopentane-1-carboxamide
(1S,5S)-3-({3-[(4-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyridine
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-ethyl-4-{[2-(4-fluorophenyl)piperidin-1-yl]sulfonyl}piperazine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-oxocyclopentyl)acetamide
2-cyclopropyl-4-hydroxy-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}pyrimidine-5-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
1-{2-[(4-chlorophenyl)methyl]benzoyl}piperidine-4-carbonitrile
(1R,5S,6R)-3-[(4-acetamidophenyl)methyl]-N-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-benzyl-N-methyl-2-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2,3-dihydro-1H-inden-2-amine
5-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-methyl-4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)piperazine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-[3-(4-{[2-(3-phenylpiperidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
[(2S,6S)-4-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(1R,5R)-3-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
8-[1-(2-methoxyphenyl)propan-2-yl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-1H-indole
2-(2-ethoxyphenyl)-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-imidazole
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(5-methoxyfuran-2-carbonyl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-5-methoxyfuran-2-carboxamide
{[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(2,3-dihydro-1H-indol-1-yl)-2-oxoacetamide
5,7-dimethyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{3-[3-(5-acetylthiophen-3-yl)phenyl]-1H-pyrazol-1-yl}-N-methylacetamide
{4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-1,4-oxazepan-6-yl}methanol
methyl 5-(cycloheptylamino)-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyrimidin-4-yl}piperidin-4-ol
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-methoxy-4-methylbenzamide
methyl 1-[(3S,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
3-(6-methoxynaphthalene-2-carbonyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
N-[(2,3-difluorophenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide