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2,5-dimethyl-3-(4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrazine
1-({[1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-methoxy-5-methylbenzoyl)piperidine
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-9H-purine
1-{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-1,2,4-triazole
N-(oxolan-2-ylmethyl)-3-[1-(3-phenylpropyl)piperidin-4-yl]propanamide
1-benzyl-6-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-indole
3-chloro-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methoxybenzamide
2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzonitrile
(3S)-3-ethyl-4-[5-(ethylsulfanyl)thiophene-2-carbonyl]morpholine
N-(isoquinolin-5-ylmethyl)-5-methoxy-N-methyl-1H-indazole-3-carboxamide
N-(2-methylpropyl)-1-[1-(1-propylpiperidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-N-ethyl-4-{[(4-methylphenyl)amino]methyl}benzamide
2-(ethylsulfanyl)-5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}pyrimidine
methyl(propan-2-yl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
methyl 4-[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]butanoate
4-benzyl-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
methyl 3-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 2-{[3-(phenylmethanesulfonamidomethyl)piperidine-1-carbonyl]amino}acetate
1-{4-[(2-ethoxypropyl)(methyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-(3-chloro-4,5-diethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-methyl-4-(2-methyl-1-benzofuran-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
8-methoxy-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(5-methylpyridin-2-yl)-1-[2-(propan-2-ylsulfanyl)ethyl]piperidin-4-ol
2-(phenoxymethyl)-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-oxazole
9-(3-hydroxy-2-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}pyridin-2-amine
9-(pyrazine-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-cyclobutyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-6-methylpyrimidin-2-amine
3-(2-aminoethyl)-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2,5,6-trimethyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidin-4-amine
5-[3-(2-ethylpiperidin-1-yl)-3-oxopropyl]-5-methylpyrrolidin-2-one
1-({4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[1-(hydroxymethyl)cyclopentyl]acetamide
3-pentyl-9-(thiophene-2-carbonyl)-3,9-diazaspiro[5.5]undecane
2-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
N-[1-(3-chlorophenyl)cyclopropyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
ethyl 1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
8-[1-(benzenesulfonyl)cyclopropanecarbonyl]-1-oxa-8-azaspiro[4.5]decane
2-ethyl-9-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-3-(2,6-difluoro-3-methylbenzoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropyl-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N2-benzyl-N2,7,7-trimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine