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6-(2-fluoro-3-methoxyphenyl)-2-methyl-1H-imidazo[4,5-b]pyridine
(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-oxazepan-6-yl)methanol
3-(azetidine-1-carbonyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]benzene-1-sulfonamide
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
4-[6-(hydroxymethyl)pyridine-2-carbonyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
1-cyclopentyl-3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]urea
2-[(3-fluorophenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1R,2S,6R,7S)-4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-4-azatricyclo[5.2.2.02,6]undecane
(3S,4S)-1-[3-(N-methylmethanesulfonamido)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methylphenol
2-(2,2-diphenylethyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]morpholine
3-[2-(morpholin-4-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-[1'-(2,5-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
{1-[1-(2-methoxyphenyl)propan-2-yl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
N-[(5-methylpyrazin-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
3-methyl-N-[2-(3-methylpiperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-(cyclopropylmethyl)-4-{[(2-methylpyridin-4-yl)methyl]sulfamoyl}benzamide
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-1-methylazepane-2-carboxamide
2-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-1H-imidazole
7-propyl-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,7-diazaspiro[4.5]decan-6-one
N4-[3-(1H-imidazol-1-yl)propyl]-6-(propan-2-yloxy)pyrimidine-2,4-diamine
N3-cyclooctyl-N5-(3-methoxypropyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N,N,4-trimethyl-6-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
4-[4-(hydroxymethyl)benzoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
ethyl 1-(oxan-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1'-(2-ethylpyridine-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 5-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazol-4-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
7-(cyclohexylmethyl)-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
(1R,5R)-6-(2-methoxyethyl)-3-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
6-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}piperidin-2-one
4-(4-hydroxy-3-methoxybenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
(4S)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-methyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
6-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(propan-2-yloxy)propanamide
3-(1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(dimethylamino)ethyl]amine
5-(dimethylamino)-2-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydropyridazin-3-one
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
(4aS,8aS)-N-(3-chloro-2-ethoxyphenyl)-4a-hydroxy-decahydroisoquinoline-2-carboxamide
4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)furan-2-carboxamide
2-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3,4,7-trimethyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-indole-2-carboxamide