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8-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
(3S,7S)-5-[3-(pyridin-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-butyl-3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-(adamantan-2-ylmethyl)-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)acetamide
N2-[(6-chloropyridin-3-yl)methyl]-N4-ethylpyrimidine-2,4-diamine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(morpholin-4-yl)propyl]-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
(1R,5S,6R)-3-[4-(piperidin-1-yl)benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[2-(morpholin-4-yl)ethyl]amine
2-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
4-{1-[1-(oxan-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
6-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-2,3-dimethylquinoxaline
6-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
3-(1-{1-[1-(3-methoxyphenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
2-chloro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1H-pyrazol-1-yl)benzamide
1-benzyl-N-methyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
6-({[1-(benzenesulfonyl)piperidin-4-yl]amino}methyl)-1,4-oxazepan-6-ol
2-{2-[(quinolin-3-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-2-yl)acetamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
N,N-dimethyl-5-[({[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]carbamoyl}amino)methyl]furan-2-carboxamide
5-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
1-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
N-[2-(ethanesulfonyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-(4-acetylphenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-amino-6-(1H-indol-3-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecane
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
N-[2-(diethylamino)ethyl]-N-ethyl-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3R,4R)-3-methyl-1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
3-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)carbamoyl]amino}-N,4-dimethylbenzamide
5-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidin-2-amine
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
(3S)-3-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}azepan-2-one
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxybutan-1-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenoxy)acetamide
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(quinolin-8-yl)pyridine-3-carboxamide
3,5-dimethyl-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-1,2-oxazole-4-carboxamide
1-(piperazin-1-yl)-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-acetyl-N-[4-chloro-3-(ethylcarbamoyl)phenyl]-1,4-diazepane-1-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
3-{[(1R,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
2-{2-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[(3S,4R)-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
4-({1-[(4-fluorophenyl)methyl]-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine