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4-{[3-(6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
3-[2-(4-fluorophenyl)ethyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
4-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]-1-(4-methylphenyl)pyrrolidin-2-one
3-benzoyl-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
2-[3-(1H-indol-3-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-[5-(1H-1,2,3-benzotriazol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]acetic acid
dimethyl[(4-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1,3-thiazol-2-yl)methyl]amine
[(3R,4R)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]piperidine-3-carboxamide
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-({5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-(4-chlorophenyl)-1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methylbutan-1-one
3-(furan-2-yl)-3-({2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}formamido)propanoic acid
(1S,3R)-3-amino-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}cyclopentane-1-carboxamide
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenol
2-(5-acetylthiophen-3-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
3-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-N-(2,4,6-trimethylphenyl)propanamide
3-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
5-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methyl-1,2-dihydropyridin-2-one
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyrazine-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)(methyl)(1H-pyrazol-3-ylmethyl)amine
N-[(2R,4R,6S)-2-tert-butyl-6-(2-ethoxyphenyl)oxan-4-yl]acetamide
3-{1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}hexan-1-one
N,N-dimethyl-5-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyridin-2-amine
N-benzyl-4-cyclobutaneamido-N-(prop-2-yn-1-yl)benzamide
({6-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazin-2-yl}methyl)dimethylamine
ethyl 1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
4-(4-chlorophenyl)-1-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]butan-1-one
N-{1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-[6-(morpholin-4-yl)pyrimidin-4-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
N-(butan-2-yl)-4-oxo-N-(pyridin-4-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(4aR,7aS)-1-(2-methylpropyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
5-[5-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
(5-{[1-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
ethyl 4-[1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
9-(2-fluoro-4-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-{[3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carbonyl]amino}-1-benzothiophene-2-carboxylate
3-(diphenylmethyl)-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-5-carboxamide
1-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-2-one
N-[(3R,4R)-3-hydroxy-1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide
4-({[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]amino}methyl)hepta-1,6-dien-4-ol
5-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(3-methoxyphenyl)piperazine