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4-(cyclopropylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(cyclohex-1-en-1-yl)-1-[4-(4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
2-(1-benzothiophen-2-ylmethyl)-4-[4-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2,4-dimethoxy-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
methyl 3-[(2E)-2-methylbut-2-en-1-yl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[2-methoxy-5-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]methanol
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-[3-(methylsulfanyl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-3-(1-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-imidazol-2-yl)-1,2-dihydroquinolin-2-one
ethyl 4-[5-(cyclopentylcarbamoyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carbonyl]piperazine-1-carboxylate
dimethyl({4-methyl-5-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
5-[(2E)-but-2-en-2-yl]-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
3-(propoxymethyl)-N-[2-(trifluoromethoxy)phenyl]pyrrolidine-1-carboxamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-(5-{1-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
3-ethyl-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-butyl-N-(3-phenylprop-2-yn-1-yl)acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
1-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidin-4-ol
(3R,4S)-4-[(benzylsulfamoyl)(ethyl)amino]oxolan-3-ol
2-methyl-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenol
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-{2-[4-(2-ethylphenyl)-1H-1,2,3-triazol-1-yl]ethyl}pyrazine
1-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-3-phenylpropan-1-ol
N,6-dimethyl-2-(morpholin-4-yl)-N-(thiophen-3-ylmethyl)pyrimidin-4-amine
2-(3-chloro-4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(pyridin-4-yl)ethyl]amine
N3-butyl-1-cyclohexyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-oxo-5-phenylpentanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-(2-methylphenyl)-3-oxo-3-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-4-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-1,2-dihydropyridin-2-one
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
2-ethyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]pyrimidine-5-carboxamide
3-(hydroxymethyl)-1-({3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl}methyl)piperidin-3-ol
2-[1-(furan-3-ylmethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-yl]ethan-1-ol
3-({[(5-chloro-2-ethoxyphenyl)methyl](methyl)amino}methyl)piperidin-3-ol
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
6-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-2-carbonitrile
(2S,4R)-4-amino-N-ethyl-1-[(5-methoxy-1H-indazol-3-yl)methyl]pyrrolidine-2-carboxamide
4-acetyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
2-(3-methoxyphenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
7-cyclohexyl-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
8-pentanoyl-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 4-{[4-(5-cyclopropaneamido-1H-pyrazol-1-yl)piperidin-1-yl]methyl}benzoate