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2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-2-ylsulfanyl)propanamide
butyl 7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
1-({5-[4-(ethylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
2-(4-{[methyl(5-methylpyrimidin-2-yl)amino]methyl}piperidin-1-yl)ethan-1-ol
6-(2,5-dimethylfuran-3-yl)-N-(4-hydroxybutyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-amino-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-6-(pyridin-2-yl)pyridine-3-carbonitrile
N-{2-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-fluorobenzamide
N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-3,6-dimethyl-1-benzofuran-2-carboxamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
(1S,5R)-3-acetyl-N-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
1-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}morpholine
N-[(3R,4S)-1-(2-carbamoylethyl)-4-cyclopropylpyrrolidin-3-yl]-4-chloro-3-fluorobenzamide
(3S,7S)-5-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(pyridin-3-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-5-carboxamide
3-(1H-1,2,4-triazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
1'-[(3-fluoro-4-methoxyphenyl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-benzyl-5-(1H-indole-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2R)-1-{2-[(prop-2-en-1-yl)amino]benzoyl}pyrrolidine-2-carboxamide
methyl 4-(5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
5-(cyclopentylmethyl)-4-(3,5-dimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(cyclohexylmethyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}piperidin-2-one
3-[3-({[2-(azepan-1-yl)ethyl](ethyl)carbamoyl}amino)phenyl]-N-methylpropanamide
3-(dimethyl-1,2-oxazol-4-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
1-(2-aminopyrimidin-4-yl)-4-(1H-1,3-benzodiazol-1-yl)piperidine-4-carboxylic acid
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
3-(4-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(1R,5S)-3-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane
(4aS,7aR)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
{[5-(4-fluoro-2-methoxyphenyl)-2-methoxyphenyl]methyl}(methyl)amine
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-cyclopropylquinoline-4-carboxamide
2-amino-4-[2-(benzylamino)pyrimidin-5-yl]-6-cyclopropylpyridine-3-carbonitrile
1-tert-butyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
[4-methyl-5-({1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-4H-1,2,4-triazol-3-yl]methanol
2-(4-{[(5-amino-1,3,4-thiadiazol-2-yl)methyl]amino}-6-methylpyrimidin-2-yl)phenol
3-[3-ethyl-5-(3-methyl-4-oxo-3,4-dihydroquinazolin-7-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-[(4-methoxyphenyl)methyl]-1-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-5-one
1-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one