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N-[2-(5-methyl-4-{[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
N-cyclopentyl-1-methyl-5-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-chlorophenyl)-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclopropane-1-carboxamide
N-[(4-fluorophenyl)methyl]-3-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}propanamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-[1'-(5-ethylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(2S,4R)-4-amino-1-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(cyclopropylmethyl)-1-({[(2-fluorophenyl)methyl]carbamoyl}methyl)piperidine-3-carboxylic acid
7-[4-(4-ethoxy-3-methylphenyl)butanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
5-fluoro-2-(5-{spiro[2.3]hexane-1-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)-1H-1,3-benzodiazole
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-[3-cyclopentyl-5-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-[5-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)furan-2-yl]benzonitrile
2-{3-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
methyl 2-(1-{[4-(1H-pyrazol-5-yl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
methyl (2S,4R)-1-(3-phenylpropyl)-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
7-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N3-methyl-1-(3-methylbutyl)-N5-[(4-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2-dihydrophthalazin-1-one
2-[4-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-[3-(1H-imidazol-5-yl)phenyl]-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2-dimethyl-2-(thiophen-2-ylformamido)propanamide
3-(1H-imidazol-1-ylmethyl)-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]propanamide
1-(4-fluorophenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]cyclopropane-1-carboxamide
methyl 2-[butyl(methyl)sulfamoyl]-6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-ethylpiperazine
methyl 1-[(3R,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-[(4-phenylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 3-methoxy-5-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]benzoate
8-(2,6,8-trimethylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
(2R,4S)-4-hydroxy-1-[(8-methoxyquinolin-2-yl)methyl]piperidine-2-carboxylic acid
3-({4-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-methyl-2-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(cyclohexylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
6-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(1-phenylcyclopentyl)methyl]acetamide
N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
(3R,4R)-3-cyclopropyl-N-[(2-fluorophenyl)methyl]-3-hydroxy-4-methylpyrrolidine-1-carboxamide
2-[1-({1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(3S,4S)-1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-[(4-fluorophenyl)methyl]-3-(pentan-3-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methylphenyl)methyl]piperidine
methyl 4-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)benzoate