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(1R,2R)-2-{ethyl[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]amino}cyclohexan-1-ol
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(1-propyl-1H-1,2,3-triazol-4-yl)benzamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(9H-purin-6-yl)piperidin-4-amine
9-(4-methylpyrimidine-5-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
4,6-dimethyl-2-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2-dihydropyridine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
2-methoxy-N-[1-(2-phenylethyl)-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
methyl[(3-methylpyridin-4-yl)methyl]{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amine
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1H-imidazol-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
2-methoxy-1-[1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5-methoxyfuran-2-carboxamide
(3S,4S)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
5-chloro-N-cyclopropyl-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
2-(dimethylamino)-2-(thianthren-1-yl)acetic acid
(1R,5S)-N-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-{[4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]methyl}phenol
2-[(3,5-difluorophenyl)methyl]-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1,2-oxazole-3-carboxamide
8-(dimethoxy-1,3,5-triazin-2-yl)quinoline
5-fluoro-N4-methyl-N2-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyrimidine-2,4-diamine
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-cyclopentyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[4-(1-ethyl-1H-imidazol-5-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
N-(3,3-dimethyl-2-oxobutyl)-4-methylnaphthalene-1-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(4-fluorophenyl)butan-1-one
(1R,3S,5S)-8-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-8-azabicyclo[3.2.1]octan-3-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}methanesulfonamide
1-(furan-3-ylmethyl)-4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazole
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
(2S,4R)-1-benzyl-N-(2-methoxyethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidine
N-(2-methylpropyl)-1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-[(2,3-dichloro-4-methylphenyl)methyl]-1-(4-methoxyphenyl)piperazin-2-one
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopentyl-2-{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]amino}propanamide
(2S)-2-amino-3-hydroxy-1-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
2-chloro-N-[2-(pyridine-3-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2,3-dimethyl-7-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
(2E)-4-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-2-enamide
3-({[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-(furan-2-yl)-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-imidazole
3-(1-{[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
(1R,5S,8R)-3-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol