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2-methyl-9-(5-propyl-1,3,4-oxadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2-hydroxy-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzoic acid
4-(1,4-diazepane-1-carbonyl)-N-[(3-methylthiophen-2-yl)methyl]aniline
N-benzyl-N-methyl-3-(4-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(2S,4S)-N-ethyl-4-[2-methyl-5-(propan-2-yl)furan-3-amido]-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}cyclopentanecarboxamide
(3S,4S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
1-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-cyclopropyl-9-(4-fluoro-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
6,8-dimethyl-3-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-{1,4-bis[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[6-(dimethylcarbamoyl)pyrazin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-N-(2,5-dimethoxyphenyl)-3-(dimethylamino)-4-propylpyrrolidine-1-carboxamide
3-(5-methyl-4H-1,2,4-triazol-3-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
N-ethyl-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
methyl 4-({3-[1-(oxan-4-ylformamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
2-(1-benzyl-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
2-amino-N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(5-oxopyrrolidin-2-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2-[3-(trifluoromethyl)phenyl]acetamide
1-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2H-1,3-benzodioxole-5-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(8-methoxy-2H-chromen-3-yl)methyl]methylamine
2-(1H-indol-3-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
3-cyclopropyl-4-(2,3-dichlorophenyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-cyclohexyl-1,4-diazepane
2-cyclopropyl-8-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-3-(2-oxooxolan-3-yl)-N-(thiophen-3-ylmethyl)propanamide
(1S,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-[2-(3-methoxyphenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-({4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
4-methyl-5-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H-pyrazolo[3,4-d]imidazol-5-yl)-1H-imidazole
2-cyclohexyl-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1H-pyrazol-1-yl)propan-2-yl]amine
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-5-methylphenol
5-[(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole