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1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
7-(7-fluoro-4-methylquinolin-2-yl)-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-chloro-N-cyclopropyl-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-3-phenylpropan-2-ol
5-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}isoquinoline
N,N-dimethyl-5-[(1-oxo-1,2-dihydrophthalazin-2-yl)methyl]furan-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-phenylpyrimidine-5-carboxamide
2-(4-{[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
5-acetamido-2-ethyl-1-(pyridin-3-ylmethyl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,3-dimethylpiperazin-2-one
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(2-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1,1-dioxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
1-cyclopentyl-4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
(2S,4S)-4-amino-N-methyl-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
methyl 1-{7-acetamido-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazole-5-carbonyl}piperidine-2-carboxylate
N-[(1S)-1-{3-cyclopropyl-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-3-(methylsulfanyl)propyl]acetamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1S,5R)-3-benzyl-N-(furan-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[4-(6-methoxypyridin-2-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-(carbamoylmethyl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]piperidine-4-carboxamide
1-(3-chloro-2-methylbenzenesulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1,3-dimethyl-N-[(3R,5S)-5-(methylcarbamoyl)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(3-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-oxoazepan-3-yl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-5-(1H-imidazol-2-yl)thiophene-2-carboxamide
2-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
5-ethyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
(3S,4S)-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-methyl-N-[3-(oxolan-2-yl)propyl]piperidin-4-amine
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
3-(1-benzothiophen-3-yl)-1-methyl-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
4-(2-fluorophenoxy)-1-(6-methoxypyrimidin-4-yl)piperidine-4-carboxylic acid
7-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-ethyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{5-methyl-3-[(phenylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
2-ethyl-5-{5-[(5-fluoro-2-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
N-(propan-2-yl)-2-[4-(2,3,5,6-tetramethylbenzoyl)piperazin-1-yl]acetamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(4-methylphenyl)piperidine-1-carboxamide
2-methyl-5-{[4-(thiomorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}-1,3-benzothiazole
4-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-1,3-oxazole-5-carboxamide
2-[(2S,5R)-2,5-dimethylpiperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
3-(3-methoxybenzoyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one