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(3S,4S)-1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(morpholin-4-yl)pyrrolidin-3-ol
4-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-6-methoxypyrimidin-2-amine
2-{3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
4-hydroxy-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
3-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
3-amino-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
2-[2-(dimethylamino)ethyl]-9-[4-(dimethylamino)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-(5-chloro-2-methylphenyl)-3-oxo-3-[3-oxo-2-(propan-2-yl)piperazin-1-yl]propanamide
2-(3-chloro-4-hydroxyphenyl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
1-methyl-1-(2-oxo-2-{3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)urea
N-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
6-cyclopentyl-1-methyl-N-[1-(pyridin-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
1-[(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-2-oxo-2-(pyrrolidin-1-yl)acetamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-[2-(cyclopropylmethyl)-4-{[2-(1H-pyrazol-4-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
2-(1-ethylpiperidin-4-yl)-N-[1-(4-hydroxyphenyl)propyl]acetamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(3-methoxy-4-propoxyphenyl)ethyl]amine
N-cyclopentyl-N'-[(3-ethoxy-4-methoxyphenyl)methyl]-N'-methylbutanediamide
3-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-(6-methylpyrimidin-4-yl)piperidin-4-amine
[(3R,4S)-1-[(3-chlorophenyl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-methanesulfonyl-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
methyl 2-{2-[3-(morpholin-4-yl)-3-oxopropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanoate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,5-dimethyl-3-phenyl-1,2-oxazole-4-carboxamide
{2-[2-methoxy-6-(4-phenyl-1H-imidazol-5-yl)phenoxy]ethyl}dimethylamine
2-[4-(butan-2-yloxy)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(methylsulfanyl)propan-1-one
1-{2-[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-1H-1,2,3-triazole
N,6-dimethyl-N-[4-(morpholin-4-yl)butyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(1R,7S)-N-methyl-3-(3-methylbutyl)-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-methoxy-2-({2-methyl-2,8-diazaspiro[4.5]decan-8-yl}methyl)phenol
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]acetamide
4-[({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
N-[(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
4-(4-chlorobenzoyl)-1-phenylpiperazin-2-one
4-(4-fluoro-2-methylphenoxy)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-4-carboxylic acid
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(3-hydroxypropanoyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
5-{[(2,4-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2,3-dihydro-1H-indene-5-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-{1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(3,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(6-methylpyridin-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2,5,6-trimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine