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2-(adamantan-1-yl)-4-hydroxy-N-(2-hydroxyethyl)-N-methylpyrimidine-5-carboxamide
1-methanesulfonyl-3-(2-phenylethyl)piperidine
N-cyclopropyl-4-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperazine-2-carboxamide
4-{[1-(butan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(1-butyl-1H-imidazol-2-yl)-N-[(1R)-1-(4-fluorophenyl)ethyl]piperidine-1-carboxamide
3-(3-hydroxybutyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
8-(2-methylquinolin-4-yl)-1-oxa-8-azaspiro[4.5]decane
methyl 2-[({3-hydroxy-1-[(3-methylphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]acetate
8-chloro-2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}quinoline
6,7-dimethoxy-2-[3-(1H-pyrazol-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
5-benzyl-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methoxyphenyl)propanamide
(3S,4R)-1-(4-hydroxy-1-methylpiperidine-4-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-{2-[(2-methoxyethyl)amino]ethyl}-1-[2-(2-methoxyphenyl)ethyl]pyrrolidin-2-one
4-{4-phenyl-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-imidazol-5-yl}benzonitrile
4-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
{3-[(3-chlorophenyl)methyl]-1-(1-phenylpiperidin-4-yl)piperidin-3-yl}methanol
2-[1-benzyl-4-(isoquinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
3-chloro-N-(cyclobutylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
2-(4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
2-cyclohexyl-5-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine-3-carboxamide
N-(2-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)oxolane-2-carboxamide
N-{[1-(5-chloro-2-methoxybenzenesulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
(3S,4R)-3-ethyl-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4-methylpiperidin-4-ol
1-[4-(benzyloxy)piperidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
5-(1H-indol-1-ylmethyl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
3-[1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)piperidin-3-yl]benzoic acid
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
2-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-6-methylquinolin-4-ol
N-[(2R)-oxolan-2-ylmethyl]-3-propyl-1H-pyrazole-5-carboxamide
4-{[3-(naphthalen-2-yl)phenyl]methyl}piperazine-1-sulfonamide
6-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(4-fluorophenyl)methyl]-N-propylpyrazine-2-carboxamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine-4-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-propyl-1,2,3-thiadiazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperazine
2-methyl-4-{5-[({[1-(2-methylpropyl)piperidin-4-yl]methyl}amino)methyl]thiophen-2-yl}but-3-yn-2-ol
6-cyclopentyl-2-methoxy-3-[({thieno[3,2-d]pyrimidin-4-yl}amino)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
[(6-chloropyridin-3-yl)methyl](methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
3-cyclopentyl-1-[(4-fluorophenyl)methyl]-5-methyl-1H-1,2,4-triazole
N-(2-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
1-(2-methyl-1-benzofuran-5-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-(2-{[2-(cyclohexylsulfanyl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-[1-(4-methoxyphenyl)propyl]-N,1-dimethyl-3-phenyl-1H-pyrazole-5-carboxamide
3-ethyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide