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N-[3-(4-methoxyphenyl)propyl]-6-(4-methyl-3-oxopiperazin-1-yl)pyridine-3-carboxamide
N-cyclopentyl-2-(2-methoxyethoxy)-N-(3-phenylprop-2-yn-1-yl)acetamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,5-dimethylpyrimidin-4-amine
2-cyclopentyl-9-[(5-hydroxy-2-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
4-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl]pyridine
7-cyclohexyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(furan-2-ylmethyl)-N-(2-methylpropyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl 5-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N3-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)piperidine-1,3-dicarboxamide
[(2S,6S)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
6-cyano-N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyridine-3-carboxamide
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N1-[3-(2-methoxyacetamido)-2-methylphenyl]piperidine-1,3-dicarboxamide
N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-2-[4-(pyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
N-({7-[3-(2-fluorophenyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
4-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
8-[3-(ethanesulfinyl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(2,3-dihydro-1H-inden-2-yl)-1,2-oxazole-3-carboxamide
4-cyclobutyl-6-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
7-[(3,4-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-methyl-2-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
5-amino-3-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-5-propylpyrimidine
1-(1-methyl-5-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-cyclopropyl-1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-(2-methoxyethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
6-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyrazine-2-carboxamide
N-[(2S)-1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methyl-1-oxopentan-2-yl]acetamide
2-(6-hydroxypyrimidin-4-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-ylmethyl]-6,8-dimethylquinolin-4-ol
1-{4-[(2-hydroxybutyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
4-{3-[2-(2-hydroxyethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-hydroxypropan-1-one
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-[5-(propan-2-yl)pyrimidin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(thiophen-2-yl)acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
(4-{5-[1-(pyrrolidin-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
1-[(3,5-dimethylphenyl)methyl]-4-[2-(propan-2-ylsulfanyl)acetyl]piperazin-2-one
4-[(1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)methyl]morpholine
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole
3-{5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazole