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2-{[5-(1H-pyrazol-4-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2,6-dimethyl-N-(1-methyl-6-oxopiperidin-3-yl)quinoline-4-carboxamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
2-cyclopropanecarbonyl-8-[(2-ethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(3,3-dimethylbutanamido)ethyl]-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-5-methylthiophene-2-carboxamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
8-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
3-(4-chloro-1H-pyrazol-1-yl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[1-(adamantane-1-carbonyl)azetidin-3-yl]pyridine
1-cyclohexyl-3-(oxolan-3-yl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-cyclopropanecarbonyl-8-(2-phenoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{4-[6-amino-5-cyano-4-(4-hydroxy-3-methylphenyl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
N-[(1S)-2,3-dihydro-1H-inden-1-yl]-4-(4-methylphenoxy)piperidine-4-carboxamide
1-methyl-3-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
1-[3-(3-fluorophenyl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
[(3R,4R)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-(4-{[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
ethyl 5-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)carbamoyl)-2,4-dimethyl-1H-pyrrole-3-carboxylate
6-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]pyrimidine-2,4-diamine
N-(oxolan-2-ylmethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
2-{4-[2-(2,5-dimethyl-1H-pyrrol-1-yl)ethyl]piperazin-1-yl}-N,N,5-trimethylpyrimidin-4-amine
3-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1λ6-thiolane-1,1-dione
4-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)morpholine
2-amino-N-[4-(3-chloro-4-methoxyphenyl)-2-fluorophenyl]acetamide
2-(2,4-difluorophenyl)-2-{[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]formamido}acetic acid
2-ethyl-8-[1-(2-methoxyacetyl)-4-methylpiperazine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
({6-[(3-fluorophenyl)methoxy]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
6-[2-(naphthalen-2-yl)acetyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
[3-(2-methoxyethyl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methanol
methyl N-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)carbamate
4-(1H-imidazol-1-ylmethyl)-1-[(4-methanesulfonylphenyl)methyl]piperidin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({7-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
4-(4-methylpiperazin-1-yl)-6-(5-methylpyridin-3-yl)pyrimidin-2-amine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
5-butyl-4-(4-methoxy-2-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]cyclopentane-1-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-benzyl-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
3-tert-butyl-1-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
1-(4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one