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N,N,4,5-tetramethyl-6-[4-(1H-1,2,3,4-tetrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-chloro-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridin-2-amine
2-methyl-5-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}pyrazine
1,3-dimethyl-6-(pyridin-4-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)-N-methylbutanamide
(3R,4S)-4-(3-methoxyphenyl)-1-(oxan-4-yl)pyrrolidin-3-amine
N-[3-(pyridin-3-yl)propyl]-2-[(thiophen-2-ylmethyl)amino]benzamide
1-methyl-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2R,6S)-4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
1-[2-(piperazin-1-yl)ethyl]-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-phenylpentanamide
methyl 4-[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]benzoate
6-tert-butyl-3-(pyrrolidin-3-yl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(4aS,8aS)-2-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-decahydroisoquinolin-4a-ol
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-(4-methylpiperazine-1-carbonyl)-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrazine
6-{1-[(2-methoxyquinolin-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(thiophen-3-ylmethyl)amine
8-[(2,5-difluorophenyl)methyl]-3-[3-(dimethylamino)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-1-ethyl-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6,7-dimethoxy-2-[3-(1H-pyrazol-5-yl)phenyl]quinazolin-4-amine
N-{3-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
3-(methoxymethyl)-N-[4-(3-methoxyphenoxy)phenyl]piperidine-1-carboxamide
1-benzyl-8-[(3-hydroxyphenyl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(2-phenylethyl)acetamide
3,5,7-trimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-indole-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-{1-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-4-(piperidin-1-yl)butanamide
4,4,4-trifluoro-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]butan-1-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]acetamide
3-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
4-oxo-5-phenoxy-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,4-dihydropyridine-3-carboxylic acid
3-{4-[(dimethylamino)methyl]phenyl}-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-methyl-4-(3-phenoxypropanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}quinolin-8-ol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
N-{4-[(2-methoxyethyl)carbamoyl]phenyl}-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,5-dimethyl-3-phenyl-1,2-oxazole-4-carboxamide
2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carbonitrile
3-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]-N-(pyridin-3-yl)propanamide
2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
4-[(4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}furan-2-yl)methyl]morpholine
2-(3,5-dimethyl-4-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
2-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenyl]-6-phenyl-3,4-dihydropyrimidin-4-one