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2-[(3,4-difluorophenyl)methyl]-8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-acetamidoacetamide
4-(5-propylpyrimidin-2-yl)benzamide
ethyl 1-[(8-fluoroquinolin-2-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
5-[4-fluoro-3-(hydroxymethyl)phenyl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{5-[(3-aminoazepan-1-yl)methyl]pyrimidin-2-yl}benzenesulfonamide
1-{1-[2-(1H-imidazol-2-yl)benzoyl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[({2-[(4-methoxyphenyl)sulfanyl]ethyl}amino)methyl]pyrrolidin-3-ol
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
3-[({[4-(aminomethyl)phenyl]methyl}amino)methyl]-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}piperidin-4-amine
(2S,4R)-4-{4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylpyrrolidine-2-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(2,3-dihydro-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-methoxy-6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidine
(3S,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
2-ethoxy-5-(2-{[(2S)-2-hydroxypropyl]amino}pyrimidin-4-yl)benzoic acid
N-[(3-fluoro-2-methoxyphenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
4-(2,4-dioxoimidazolidin-1-yl)-N-[3-(pyridin-3-yloxy)propyl]benzamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
N'-(3-ethylphenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]butanediamide
(2S,4R)-1-benzyl-N,N-diethyl-4-{[(2-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(9H-purin-6-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
(2S,4R)-4-amino-1-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-[1-(naphthalene-2-carbonyl)piperidin-4-yl]ethyl]cyclobutanecarboxamide
N-cyclopropyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
4-[4-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
1-(1-benzothiophene-5-carbonyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-phenyl-1H-imidazol-1-yl)acetamide
2-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5-methyl-1,3,4-oxadiazol-2-amine
3-chloro-N,2-dimethyl-N-(pyrazin-2-ylmethyl)benzamide
(4aS,7aR)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(4S,4aS,8aS)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
({4-ethyl-5-[1-(oxane-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-{[4-(3-chloro-5-methylpyridin-2-yl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
1-[3-(3-chlorophenyl)phenyl]-3-[2-(4-methylpiperazin-1-yl)propyl]urea
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
4-(4-ethoxyphenyl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
(4aR,7aS)-1-(2-methoxyacetyl)-4-{2-[methyl(phenyl)amino]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-methyl-1-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propan-2-yl}-1,2,3,4-tetrahydroisoquinoline
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
2-[1-(cyclohexylmethyl)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidine-2-carboxylic acid
3-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{1'-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-oxo-4-phenylbutanamide