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1-cyclopentyl-4-[5-(3,4-dimethylphenyl)-4-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
1-(3-fluoro-4-methylbenzoyl)-2-(3-methoxypropyl)piperidine
1-(2-methoxyethyl)-3,8-bis(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
[3-(3-methylbut-2-en-1-yl)-1-(morpholine-4-carbonyl)piperidin-3-yl]methanol
{3-[(3-chlorophenyl)methyl]-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl}methanol
N-[(3-methylphenyl)methyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
5-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-ol
4,5-dimethyl 1-[(3S,5S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-[3-(1H-imidazol-1-yl)propyl]-4,6-dimethoxypyrimidine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-(pyridine-3-sulfonyl)piperidin-3-amine
2-cyano-N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]benzamide
8-[2-(morpholin-4-yl)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(morpholin-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
(3S,4R)-4-(hydroxymethyl)-1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-(6-methoxypyridin-3-yl)acetic acid
5-cyano-N,4-dimethyl-6-oxo-N-[(4-phenoxyphenyl)methyl]-1,6-dihydropyridine-3-carboxamide
N,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]quinoline-4-carboxamide
methyl[(4-{2-[4-(3-methylthiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](quinolin-6-ylmethyl)amine
5-(oxolane-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
N-{2-[4-(quinolin-4-ylmethyl)morpholin-2-yl]ethyl}methanesulfonamide
5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-benzoyl-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-tert-butyl-4-hydroxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
(4aS,8aR)-6-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
4-[2-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1-(propan-2-yl)-1H-pyrazole
2-(dimethylamino)-N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]acetamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenylpiperazine
1-{1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}pyrrolidin-2-one
5-[(1-benzothiophen-2-ylmethyl)(methyl)amino]-1-[(4-methoxyphenyl)methyl]azepan-2-one
3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylamino)pentanamide
4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carbaldehyde
3-(4-chlorophenyl)-N-ethyl-3-phenylpropanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-{[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indazole
3-[(2R,3R,6R)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[5-(methoxymethyl)furan-2-carbonyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(piperidin-3-ylmethyl)amine
1-cyclopentyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(3S,4R)-1-{[(1,3-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N,5-dimethyl-N-(quinolin-5-ylmethyl)-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
N-[4-(4-ethenylbenzamido)phenyl]-5-methylfuran-2-carboxamide