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1-methanesulfonyl-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-methyl-4-{4-[1-(2-methylpropyl)piperidin-4-yl]piperazin-1-yl}-6-propylpyrimidine
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(oxolane-2-carbonyl)piperazin-1-yl]acetamide
4-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-(4-methoxy-3-methylphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
N-{1-[4-(pyridin-4-yl)pyrimidin-2-yl]pyrrolidin-3-yl}acetamide
6-methoxy-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[3-(1H-imidazol-1-yl)propyl]-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
ethyl 4-[(2-chlorophenyl)methyl]-1-(2-methylfuran-3-carbonyl)piperidine-4-carboxylate
1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(3-methylbut-2-en-1-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-chlorophenyl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
methyl 1-{9-methoxy-7-oxo-3-propyl-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
7-(6,7-dimethoxy-4-methylquinolin-2-yl)-4-(furan-2-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[2-(1H-pyrazol-1-yl)phenyl]methyl})amine
2-[3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenyl]-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-N-(2-methylpropyl)acetamide
4-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-3-yl}morpholine
2-{4-[2-(3-chlorophenyl)-2-hydroxyacetyl]piperazin-1-yl}-N-ethylacetamide
(4aS,7aR)-N,N-dimethyl-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
N-(diphenylmethyl)-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-2-(oxan-2-ylmethoxy)-N-[2-(pyridin-4-yl)ethyl]acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-imidazole-2-carboxamide
(3R,9R)-11-(3-methylbutyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-2,4-dimethylpyrimidine
3-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-4-methylpyridine
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
3-{[4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
8-[2-(4-methylphenoxy)ethanesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(methylsulfamoyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-(2-methyl-4-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]carbamoyl}phenyl)furan-2-carboxamide
(3S,5R)-1-[(3-methylphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
4-chloro-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-{3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-oxopropyl}azepan-2-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-yl)ethan-1-one
4-acetyl-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]benzene-1-sulfonamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(4-methylpiperidine-4-carbonyl)piperidine
N-[3-(ethylcarbamoyl)-2-methylphenyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
3-(3-phenyl-1H-1,2,4-triazol-5-yl)-1,2-dihydroquinoxalin-2-one
ethyl 4-{[(1R,2S)-2-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetamido]cyclobutyl]amino}piperidine-1-carboxylate
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-ol
2-(2H-1,2,3-benzotriazol-2-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(methylamino)pyridine-4-carboxamide
N-(1-{7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide