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4-[3-(2,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-(1H-pyrazol-1-yl)pyrimidine
3-methyl-6-[5-(oxan-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-(propan-2-yl)pyrimidine-2,4-diamine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
N-ethyl-2-(4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)acetamide
(3aR,6aR)-2-acetyl-5-[(6-fluoro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-N-(propan-2-yl)piperidine-1-carboxamide
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
methyl (2S,4R)-1-[(4-fluorophenyl)methyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxylate
4-{[2-(2-hydroxyethoxy)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[3-(1H-pyrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-[4-ethoxy-3-(hydroxymethyl)phenyl]-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
5-[(methylsulfanyl)methyl]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
1-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-ethylurea
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(methylsulfanyl)propan-1-one
1-[1-(2,6-dimethoxybenzoyl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-1-[(1S)-1-(3-methylpyridin-2-yl)ethyl]urea
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-(thiophene-2-sulfonyl)piperidine
N-benzyl-3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
1-{2-hydroxy-3-[4-({[2-(4-hydroxyphenyl)ethyl]amino}methyl)-2-methoxyphenoxy]propyl}piperidin-4-ol
ethyl 1-{3-[(cyclopentylamino)methyl]-6,7-dimethoxyquinolin-2-yl}piperidine-3-carboxylate
N-[(3R,4S)-1-(2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-ethyl-9-(2-ethylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)propanamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(1H-pyrazol-1-yl)benzamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
2-(4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-1-yl)pyridine-3-carboxamide
2-(3-methoxyphenyl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)acetamide
(3R,4S)-4-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
methyl 3-(furan-3-amido)-5-[(quinolin-2-ylformamido)methyl]benzoate
1'-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
6-ethyl-4-(4-methanesulfonylpiperazine-1-carbonyl)-2-methylquinoline
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
(1R,3S)-3-(2-aminoethoxy)-7-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
1-(4-methyl-1,3-thiazole-5-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
1-[3-(4-fluorophenyl)phenyl]-N-(morpholin-2-ylmethyl)piperidin-4-amine
2-[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
1-(carbamoylmethyl)-3-[(4-fluorophenyl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(5-phenyl-1,2,4-triazin-3-yl)-1,4-diazepan-1-yl]-1,3-benzothiazole
1-(4-{4-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}phenyl)ethan-1-one
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
7-(5-chloropyridin-2-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol