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5-(3,3-diethylpyrrolidine-1-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-indole
2,2-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)oxane-4-carboxamide
1-methyl-2-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
2-cyclopropyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-hydroxy-N-methylpyrimidine-5-carboxamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-[4-({[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]imidazolidin-2-one
4-{5-[(4,5-dimethylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazole
8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(5-chloropyridin-2-yl)-4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
N-cyclopropyl-4-methoxy-3-({[2-(4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}amino)benzamide
methyl({[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})(quinolin-2-ylmethyl)amine
7-(2-cyclohexylethyl)-2-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2,7-diazaspiro[4.5]decane
2-(dimethyl-1,2-oxazol-4-yl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
N-[3-(1H-indol-1-yl)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
propan-2-yl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
(3R,4S)-4-(propan-2-yl)-1-(1H-1,2,3-triazol-4-ylmethyl)pyrrolidin-3-amine
N-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-[1-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)piperidin-3-yl]pyrrolidin-2-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2,5,7-trimethylquinoline-4-carboxamide
[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)sulfamoyl]dimethylamine
N-[(4-fluorophenyl)methyl]-2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
6-{2-ethyl-4-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}pyridine-3-carbonitrile
4-fluoro-N-({1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}methyl)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{5-[(4-{1-[(4-fluorophenyl)methyl]-4-methyl-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)methyl]thiophen-2-yl}acetamide
N-[2-(dimethylamino)ethyl]-N-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}cyclopentanamine
[2-(1H-imidazol-1-yl)ethyl](methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
methyl 1-{2-hydroxy-3-[4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-amine
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
N-{2-[cyclopentyl(methyl)amino]ethyl}-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-{[(5-methylpyrazin-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[(3R,4R)-1-(2-methoxy-5-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-[4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
dimethyl({1-[3-(6-methylpyridazin-3-yl)phenyl]ethyl})amine
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
3-methyl-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-(naphthalen-2-yloxy)propan-1-one
(3S,9aR)-8-(naphthalene-2-sulfonyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-3-ethylpiperidine-3-carboxylic acid
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(propan-2-yl)-4-[3-(pyrazin-2-yl)propanoyl]-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(furan-2-ylmethyl)(methyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
2-(1-benzothiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2,4-dichloro-3-({7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)phenol