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N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-(1H-pyrazol-4-yl)butanamide
4-{[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(2S,4R)-4-amino-N-ethyl-1-[2-(5-methylfuran-2-amido)benzoyl]pyrrolidine-2-carboxamide
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-hydroxy-1,2-oxazole-5-carboxamide
5-[(dimethylamino)methyl]-N-[3-(methylsulfanyl)propyl]furan-2-carboxamide
3-(1H-imidazol-4-yl)-2-{[5-(morpholin-4-ylmethyl)furan-3-yl]formamido}propanoic acid
2-(3-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-amine
1-{4-[2-(2-ethylphenoxy)ethyl]piperazin-1-yl}ethan-1-one
2-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-(1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}piperidin-2-yl)ethan-1-ol
4-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]piperazin-1-yl}-5-propylpyrimidine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
3-{[cyclopropyl({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}phenol
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methoxy-4-{2-[methyl({2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amino]propyl}phenol
4-({9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(2S,4R)-N-methyl-1-(pyrazine-2-carbonyl)-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
5-methyl-N-(2-methylprop-2-en-1-yl)-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(2S)-1-(3,3-diphenylpiperidin-1-yl)-1-oxopropan-2-yl]acetamide
4-[1-(3-phenylpropyl)-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(2S)-3,3-dimethyl-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}butanoic acid
N-{[3-(trifluoromethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(4aS,7aR)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-ethyl-9-[2-(methylamino)-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-chlorobenzenesulfonamido)ethyl]-1,4-dioxane-2-carboxamide
methyl 9-(cyclopentyloxy)-3-(1-methyl-1H-indole-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(dimethyl-1,2-oxazol-4-yl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carboxamide
1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
2-[4-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
9-{[4-(methylsulfanyl)phenyl]methyl}-6-oxa-9-azaspiro[4.5]decane
3-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-2-methoxypyridine
2-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]formamido}hexanamide
methyl 6-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]pyridine-2-carboxylate
N-(pyrazin-2-yl)-2-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)acetamide
(2S,4S)-4-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpyrrolidine-2-carboxylic acid
2-(methoxymethyl)-N-(1-methoxypropan-2-yl)-6-methyl-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(2-methoxyphenoxy)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
(5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)methanol
1-{2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide